SCHEMBL3706773

SCHEMBL3706773

CNC1(c2ccc(F)c(Cl)c2)CCCNC1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 15/20 0.49
SLC6A3 Q01959 13/20 0.49
SLC6A2 P23975 11/20 0.49
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
CYP2D6 P10635 2/20 0.38
KCNH2 Q12809 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3712314 0.87 SLC6A3 (0.46) SLC6A4SLC6A3SLC6A2HDAC3HDAC1
SCHEMBL3709523 0.84 HDAC3 (0.39) SLC6A4SLC6A3SLC6A2HDAC3HDAC1
SCHEMBL27734550 0.84 SLC6A3 (0.62) SLC6A4SLC6A3SLC6A2HDAC3HDAC1
SCHEMBL3718210 0.82 DRD2 (0.42) SLC6A4SLC6A3SLC6A2KCNH2
SCHEMBL3707150 0.80 SLC6A3 (0.47) SLC6A4SLC6A3SLC6A2HDAC3HDAC1
SCHEMBL3712760 0.79 SLC6A3 (0.41) SLC6A4SLC6A3SLC6A2HDAC3HDAC1
SCHEMBL3709501 0.79 HTR2C (0.42) SLC6A4SLC6A3SLC6A2HDAC6
SCHEMBL3705259 0.78 CTSD (0.37) SLC6A4SLC6A3SLC6A2HDAC3HDAC1
SCHEMBL4520209 0.77 SLC6A4 (0.46) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL3705030 0.77 SLC6A4 (0.47) SLC6A4SLC6A3SLC6A2HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2391603-A1 AROYLAMINO - AND HETEROAROYLAMINO-SUBSTITUTED PIPERIDINES AS GLYT-1 INHIBITORS F. Hoffmann-La Roche AG (CH) 2011-12-07 EP disclosed
WO-2010086251-A1 AROYLAMINO - AND HETEROAROYLAMINO-SUBSTITUTED PIPERIDINES AS GLYT-1 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-08-05 WO disclosed