SCHEMBL3705259

SCHEMBL3705259

CNC1(c2cc(F)cc(F)c2)CCCNC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.37
SLC6A3 Q01959 7/20 0.34
SLC6A4 P31645 6/20 0.34
HDAC3 O15379 2/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC2 Q92769 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34
SLC6A2 P23975 4/20 0.33
CHRNA1 P02708 1/20 0.33
CHRNG P07510 1/20 0.33
CHRNB1 P11230 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA4 P43681 1/20 0.33
CHRND Q07001 1/20 0.33
SLC6A9 P48067 1/20 0.33
USP2 O75604 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3705030 0.86 SLC6A4 (0.47) CTSDSLC6A3SLC6A4HDAC3HDAC1
SCHEMBL3712760 0.85 SLC6A3 (0.41) SLC6A3SLC6A4HDAC3HDAC1HDAC2
SCHEMBL3712314 0.81 SLC6A3 (0.46) CTSDSLC6A3SLC6A4HDAC3HDAC1
SCHEMBL3709523 0.79 HDAC3 (0.39) CTSDSLC6A3SLC6A4HDAC3HDAC1
SCHEMBL3707243 0.78 OPRM1 (0.49) SLC6A9USP2ALDH1A1CYP3A4OPRM1
SCHEMBL3706773 0.78 SLC6A4 (0.49) SLC6A3SLC6A4HDAC3HDAC1HDAC2
SCHEMBL3709950 0.77 SLC6A2 (0.36) SLC6A3SLC6A4HDAC3HDAC1HDAC2
SCHEMBL3711236 0.77 HDAC6 (0.36) SLC6A3SLC6A4HDAC3HDAC1HDAC2
SCHEMBL3713554 0.77 OPRM1 (0.37) SLC6A3SLC6A4HDAC3HDAC1HDAC2
SCHEMBL3718210 0.75 DRD2 (0.42) SLC6A3SLC6A4SLC6A2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2391603-A1 AROYLAMINO - AND HETEROAROYLAMINO-SUBSTITUTED PIPERIDINES AS GLYT-1 INHIBITORS F. Hoffmann-La Roche AG (CH) 2011-12-07 EP disclosed
WO-2010086251-A1 AROYLAMINO - AND HETEROAROYLAMINO-SUBSTITUTED PIPERIDINES AS GLYT-1 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-08-05 WO disclosed