SCHEMBL3707175

SCHEMBL3707175

CNC(=O)OCc1cc(Sc2cccc(F)c2)n(-c2cccnc2F)n1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 5/20 0.33
GRM5 P41594 3/20 0.33
CA2 P00918 2/20 0.32
CA4 P22748 2/20 0.32
MAPT P10636 2/20 0.32
TP53 P04637 1/20 0.32
TOP2A P11388 1/20 0.32
TOP2B Q02880 1/20 0.32
NTRK1 P04629 1/20 0.32
HDAC1 Q13547 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HDAC5 Q9UQL6 1/20 0.31
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3703976 0.81 NOTUM (0.33) SLC6A9GRM5
SCHEMBL4130901 0.80 TP53 (0.34) SLC6A9CA2CA4MAPTTP53
SCHEMBL4130894 0.80 SLC6A9 (0.36) SLC6A9CA2CA4MAPTTP53
SCHEMBL3693917 0.79 RIPK1 (0.32) MAPTTOP2ATOP2BHTT
SCHEMBL3701560 0.79 THRB (0.46) MAPTTP53LMNAHTT
SCHEMBL3805129 0.78 HTR2C (0.45) SLC6A9MAPTTP53HDAC1HDAC8
SCHEMBL16333316 0.76 KMT2A (0.36) SLC6A9MAPTLMNAHTTL3MBTL1
SCHEMBL3709000 0.75 SLC16A3 (0.37) TOP2ATOP2B
SCHEMBL3698799 0.73 SLC16A3 (0.40) TOP2ATOP2B
SCHEMBL3697121 0.73 NOTUM (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed