SCHEMBL3707271

SCHEMBL3707271

CCOC(=O)N(c1ccccc1Cl)c1c(C)noc1-c1cccc(-c2cncc(C(=O)O)c2)c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.38
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
IP6K1 Q92551 3/20 0.35
IP6K3 Q96PC2 3/20 0.35
IP6K2 Q9UHH9 3/20 0.35
ADRB2 P07550 1/20 0.34
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
NR1H4 Q96RI1 5/20 0.33
DUSP3 P51452 3/20 0.33
CTSA P10619 1/20 0.33
LIFR P42702 1/20 0.33
PTPN1 P18031 1/20 0.33
CHRNA7 P36544 1/20 0.33
BRD4 O60885 1/20 0.32
BRD2 P25440 1/20 0.32
CREBBP Q92793 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3712570 0.93 CYP2C9 (0.36) CYP2C9CYP2C19IP6K1IP6K3IP6K2
SCHEMBL3708502 0.92 IP6K1 (0.40) IP6K1IP6K3IP6K2NR1H4DUSP3
SCHEMBL3702769 0.92 S1PR1 (0.38) PDE4BNR1H4CTSACHRNA7
SCHEMBL3705512 0.89 LPAR1 (0.39) PDE4BNR1H4
SCHEMBL2336147 0.88 NR1H4 (0.42) IP6K1IP6K3IP6K2NR1H4DUSP3
SCHEMBL3714488 0.87 L3MBTL1 (0.34) CYP2C9CYP2C19
SCHEMBL3705734 0.86 KMO (0.39) IP6K1IP6K3IP6K2NR1H4LIFR
SCHEMBL3714395 0.85 NR1H4 (0.40) NR1H4
SCHEMBL3707761 0.85 DUSP3 (0.35) CYP2C9NR1H4DUSP3CTSAPTPN1
SCHEMBL3707635 0.84 CTSA (0.35) PDE4BADRB2ADRB1ADRB3CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010077882-A2 ANTAGONISTS OF LYSOPHOSPHATIDIC ACID RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2010-07-08 WO claimed
WO-2010077882-A2 ANTAGONISTS OF LYSOPHOSPHATIDIC ACID RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2010-07-08 WO disclosed