SCHEMBL3708097

SCHEMBL3708097

CCOC(=O)CN(Cc1ccc(O)cc1)C(=O)CC1C(=O)N(C(Cl)Cc2ccc(Cl)cc2)CC(=O)N1CCCN1CCOCC1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.34
ALDH1A1 P00352 2/20 0.34
USP2 O75604 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
AVPR1A P37288 4/20 0.33
MDM2 Q00987 2/20 0.33
TP53 P04637 1/20 0.33
PPARG P37231 1/20 0.33
NCOR2 Q9Y618 1/20 0.33
TACR2 P21452 4/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ATM Q13315 1/20 0.32
EPHX2 P34913 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3697424 0.93 APAF1 (0.34) TSHRALDH1A1USP2NPSR1MDM2
SCHEMBL3705051 0.90 APAF1 (0.36) TSHRALDH1A1USP2NPSR1MDM2
SCHEMBL3710700 0.89 MDM2 (0.38) TSHRALDH1A1USP2MDM2TP53
SCHEMBL3695334 0.88 MDM2 (0.35) TSHRALDH1A1USP2NPSR1MDM2
SCHEMBL9101546 0.87 C5AR1 (0.39) ALDH1A1TACR2KDM4E
SCHEMBL3701950 0.85 KCNJ1 (0.36) TSHRALDH1A1USP2NPSR1MDM2
SCHEMBL3700914 0.85 TSHR (0.41) TSHRALDH1A1USP2NPSR1AVPR1A
SCHEMBL3696385 0.85 PTGS2 (0.37) ALDH1A1KDM4E
SCHEMBL3702536 0.85 APAF1 (0.42) TSHRAVPR1APPARGNCOR2TACR2
SCHEMBL3713311 0.85 PSEN1 (0.35) TSHRALDH1A1USP2NPSR1AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9040701-B2 Apaf-1 inhibitor compounds LABORATORIOS SALVAT, S.A. (ES) 2015-05-26 US disclosed
US-20120122868-A1 APAF-1 INHIBITOR COMPOUNDS LABORATORIOS SALVAT, S.A. (ES) 2012-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120122868-A1 APAF-1 INHIBITOR COMPOUNDS APAF1, API5, AIFM1 TSHR 4570/4885ALDH1A1 701/4885USP2 1336/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.