SCHEMBL3696385

SCHEMBL3696385

CCOC(=O)CN(CCc1ccc(S(N)(=O)=O)cc1)C(=O)CC1C(=O)N(C(Cl)Cc2ccc(Cl)cc2)CC(=O)N1CCCN1CCOCC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.37
CA1 P00915 5/20 0.36
CA2 P00918 5/20 0.36
CA4 P22748 3/20 0.36
CA7 P43166 3/20 0.36
MMP2 P08253 1/20 0.35
MMP3 P08254 1/20 0.35
MMP9 P14780 1/20 0.35
MMP13 P45452 1/20 0.35
APAF1 O14727 3/20 0.34
CASP3 P42574 3/20 0.34
CASP9 P55211 3/20 0.34
CYCS P99999 3/20 0.34
CA9 Q16790 3/20 0.33
ALDH1A1 P00352 2/20 0.33
CA12 O43570 2/20 0.33
TBXA2R P21731 1/20 0.33
TBXAS1 P24557 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3705051 0.94 APAF1 (0.36) MMP2MMP3MMP9MMP13APAF1
SCHEMBL3697424 0.92 APAF1 (0.34) MMP2MMP3MMP9MMP13APAF1
SCHEMBL9101546 0.91 C5AR1 (0.39) PTGS2APAF1CASP3CASP9CYCS
SCHEMBL3701950 0.90 KCNJ1 (0.36) MMP2MMP3MMP9MMP13APAF1
SCHEMBL3704033 0.89 APAF1 (0.36) CA1CA2CA4CA7APAF1
SCHEMBL3700914 0.88 TSHR (0.41) APAF1CASP3CASP9CYCSALDH1A1
SCHEMBL3705169 0.86 ALDH1A1 (0.36) APAF1CASP3CASP9CYCSALDH1A1
SCHEMBL3702485 0.86 CA12 (0.37) CA1CA2CA4APAF1CASP3
SCHEMBL3708097 0.85 TSHR (0.34) ALDH1A1KDM4E
SCHEMBL3701029 0.85 TACR2 (0.45) APAF1CASP3CASP9CYCSALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9040701-B2 Apaf-1 inhibitor compounds LABORATORIOS SALVAT, S.A. (ES) 2015-05-26 US disclosed
US-20120122868-A1 APAF-1 INHIBITOR COMPOUNDS LABORATORIOS SALVAT, S.A. (ES) 2012-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120122868-A1 APAF-1 INHIBITOR COMPOUNDS APAF1, API5, AIFM1 PTGS2 1620/4885CA1 1810/4885CA2 2622/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.