SCHEMBL3709499

SCHEMBL3709499

COC(=O)Cc1cc2ccc(C#N)cc2[nH]c1=O

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 8/20 0.49
KDM4E B2RXH2 8/20 0.47
HSD17B10 Q99714 7/20 0.47
ALDH1A1 P00352 4/20 0.47
TSHR P16473 5/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.44
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
ALOX15 P16050 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3716513 0.84 IDH1 (0.50) IDH1KDM4EHSD17B10ALDH1A1TSHR
SCHEMBL7071513 0.82 IDH1 (0.51) IDH1KDM4EHSD17B10ALDH1A1TSHR
SCHEMBL3715876 0.81 EGFR (0.53) KDM4EHSD17B10ALDH1A1TSHRMEN1
SCHEMBL7073150 0.81 KDM4E (0.63) IDH1KDM4EHSD17B10ALDH1A1TSHR
SCHEMBL8306652 0.79 KDM4E (0.59) KDM4EHSD17B10ALDH1A1TSHRMEN1
SCHEMBL3712461 0.78 KDM4E (0.47) IDH1KDM4EHSD17B10ALDH1A1TSHR
SCHEMBL3712923 0.76 KDM4E (0.51) KDM4EHSD17B10ALDH1A1TSHRMEN1
SCHEMBL30088460 0.76 HTT (0.44) KDM4EHSD17B10ALDH1A1TP53MAPT
SCHEMBL4839414 0.76 HTT (0.44) KDM4EHSD17B10ALDH1A1TP53MAPT
SCHEMBL3709826 0.74 GABRA1 (0.41) IDH1KDM4EHSD17B10ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2393806-A1 INHIBITORS OF JUN N-TERMINAL KINASE Elan Pharmaceuticals Inc. (US) 2011-12-14 EP disclosed
WO-2010091310-A1 INHIBITORS OF JUN N-TERMINAL KINASE ELAN PHARMACEUTICALS, INC. (US) 2010-08-12 WO disclosed