SCHEMBL3710087

SCHEMBL3710087

COC(=O)c1cc(NC(=O)c2ccccc2O)nc(-c2ccc(C#Cc3cccnc3)cc2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
KMT2A Q03164 5/20 0.43
MEN1 O00255 4/20 0.43
KDM4E B2RXH2 3/20 0.43
HPGD P15428 1/20 0.43
XIAP P98170 2/20 0.40
BIRC2 Q13490 2/20 0.40
CYP19A1 P11511 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
CSF1R P07333 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
LMNA P02545 1/20 0.38
THRB P10828 1/20 0.38
HTT P42858 1/20 0.38
ABCB1 P08183 1/20 0.38
ABCC1 P33527 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3711552 0.88 ALDH1A1 (0.46) ALDH1A1KMT2AMEN1KDM4EHPGD
SCHEMBL13187749 0.88 CYP19A1 (0.50) ALDH1A1KMT2AMEN1KDM4EHPGD
SCHEMBL3712830 0.87 DEGS1 (0.44) ALDH1A1CYP19A1CYP11B1CYP11B2CSF1R
SCHEMBL3712399 0.86 GRM5 (0.46) ALDH1A1CYP19A1CYP11B1CYP11B2CYP1A2
SCHEMBL3712176 0.86 GRM5 (0.42) ALDH1A1KMT2ACYP19A1CYP11B1CYP11B2
SCHEMBL3713260 0.85 CYP11B1 (0.48) CYP19A1CYP11B1CYP11B2CSF1RSMN1; SMN2
SCHEMBL3711302 0.85 RAB9A (0.49) KMT2AMEN1HPGDCYP19A1CYP11B1
SCHEMBL3713498 0.84 CYP19A1 (0.39) ALDH1A1KMT2AMEN1XIAPBIRC2
SCHEMBL3712323 0.84 CYP19A1 (0.46) ALDH1A1XIAPBIRC2CYP19A1CYP11B1
SCHEMBL3713936 0.83 ADORA3 (0.47) ALDH1A1XIAPBIRC2CYP19A1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed