SCHEMBL3712399

SCHEMBL3712399

COC(=O)c1cc(NC(C)=O)nc(-c2ccc(C#Cc3cccnc3)cc2)c1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.46
ADORA3 P0DMS8 15/20 0.45
CYP19A1 P11511 1/20 0.44
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
ADORA1 P30542 4/20 0.43
ADORA2A P29274 3/20 0.43
ADORA2B P29275 2/20 0.43
CYP1A2 P05177 1/20 0.42
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3711552 0.90 ALDH1A1 (0.46) GRM5CYP19A1CYP11B1CYP11B2ALDH1A1
SCHEMBL3712323 0.90 CYP19A1 (0.46) GRM5CYP19A1CYP11B1CYP11B2ALDH1A1
SCHEMBL3714104 0.89 ABL1 (0.41)
SCHEMBL3713936 0.89 ADORA3 (0.47) GRM5ADORA3CYP19A1CYP11B1CYP11B2
SCHEMBL3711439 0.89 ADORA1 (0.46) GRM5CYP19A1CYP11B1CYP11B2ADORA1
SCHEMBL3715718 0.88 XIAP (0.45) GRM5ADORA3CYP19A1CYP11B1CYP11B2
SCHEMBL3710834 0.88 KDM4E (0.45) GRM5CYP19A1CYP11B1CYP11B2ALDH1A1
SCHEMBL3721325 0.88 CYP19A1 (0.44) GRM5CYP19A1CYP11B1CYP11B2ALDH1A1
SCHEMBL3714356 0.88 NAMPT (0.41) GRM5CYP19A1CYP11B1CYP11B2ALDH1A1
SCHEMBL3713698 0.88 PTGES (0.42) GRM5CYP19A1CYP11B1CYP11B2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed