SCHEMBL3710958

SCHEMBL3710958

CCCN1CCN(c2ccc(N)cc2)C1=O

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.52
DRD3 P35462 6/20 0.52
CYP1A1 P04798 8/20 0.50
S1PR1 P21453 1/20 0.50
RAB9A P51151 1/20 0.46
KCNH2 Q12809 2/20 0.46
HDAC1 Q13547 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10499028 0.90 CYP1A1 (0.56) DRD2DRD3CYP1A1S1PR1RAB9A
SCHEMBL10498437 0.86 RAB9A (0.49) DRD2DRD3CYP1A1S1PR1RAB9A
SCHEMBL14698020 0.85 DRD2 (0.65) DRD2DRD3CYP1A1S1PR1RAB9A
SCHEMBL3712107 0.80 S1PR1 (0.48) DRD2DRD3CYP1A1S1PR1RAB9A
SCHEMBL14698170 0.80 CYP1A1 (0.57) DRD2DRD3CYP1A1S1PR1RAB9A
SCHEMBL10499403 0.80 CYP1A1 (0.48) DRD2DRD3CYP1A1S1PR1KCNH2
SCHEMBL3714292 0.78 DRD2 (0.61) DRD2DRD3CYP1A1HDAC1
SCHEMBL3577171 0.77 MAPT (0.47) DRD2DRD3RAB9A
SCHEMBL13666331 0.77 KDM4E (0.45) DRD2DRD3S1PR1RAB9AHDAC1
SCHEMBL4670487 0.75 DRD2 (0.45) DRD2DRD3CYP1A1S1PR1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010099518-A2 METHOD FOR MANUFACTURE OF 2-OXOIMIDAZOLIDINES THESIS CHEMISTRY, LLC (US) 2010-09-02 WO disclosed
US-4861879-A VAGINAL FUNGICIDE JANSSEN PHARMACEUTICA N.V. (BE) 1989-08-29 US disclosed
EP-0118138-B1 ((4-(4-(4-PHENYL-1-PIPERAZINYL)PHENOXYMETHYL)-1,3-DIOXOLAN-2-YL)METHYL)-1H-IMIDAZOLES AND 1H-1,2,4-TRIAZOLES JANSSEN PHARMACEUTICA N.V. (BE) 1989-06-14 EP disclosed
US-4735942-A FUNGICIDE, BACTERICIDE PARTICULARLY FOR UROGENITAL DISORDERS JANSSEN PHARMACEUTICA, N.V. (BE) 1988-04-05 US disclosed
US-4619931-A BACTERICIDES, FUNGICIDES JANSSEN PHARMACEUTICA, N.V. (BE) 1986-10-28 US disclosed
EP-0118138-A1 ((4-(4-(4-Phenyl-1-piperazinyl)phenoxymethyl)-1,3-dioxolan-2-yl)methyl)-1H-imidazoles and 1H-1,2,4-triazoles JANSSEN PHARMACEUTICA N.V. (BE) 1984-09-12 EP disclosed