SCHEMBL3713698

SCHEMBL3713698

COC(=O)c1cc(NC(=O)NC(C)C)nc(-c2ccc(C#Cc3cccnc3)cc2)c1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGES O14684 3/20 0.42
AKR1C3 P42330 2/20 0.42
CYP19A1 P11511 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
XIAP P98170 2/20 0.41
BIRC2 Q13490 2/20 0.41
ACACB O00763 1/20 0.40
ALDH1A1 P00352 1/20 0.39
GRM5 P41594 3/20 0.39
CHRM2 P08172 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
CSF1R P07333 1/20 0.37
SLC2A1 P11166 1/20 0.37
AHR P35869 1/20 0.36
ABL1 P00519 1/20 0.36
BCR P11274 1/20 0.36
SRC P12931 1/20 0.36
FFAR1 O14842 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3709347 0.89 PTGES (0.42) PTGESAKR1C3XIAPBIRC2ACACB
SCHEMBL3713936 0.89 ADORA3 (0.47) PTGESAKR1C3CYP19A1CYP11B1CYP11B2
SCHEMBL3715718 0.88 XIAP (0.45) PTGESAKR1C3CYP19A1CYP11B1CYP11B2
SCHEMBL3710834 0.88 KDM4E (0.45) CYP19A1CYP11B1CYP11B2ACACBALDH1A1
SCHEMBL3712399 0.88 GRM5 (0.46) CYP19A1CYP11B1CYP11B2ALDH1A1GRM5
SCHEMBL13188363 0.88 CYP19A1 (0.52) CYP19A1CYP11B1CYP11B2ALDH1A1SLC2A1
SCHEMBL3714104 0.87 ABL1 (0.41) ABL1
SCHEMBL3711552 0.86 ALDH1A1 (0.46) CYP19A1CYP11B1CYP11B2ALDH1A1GRM5
SCHEMBL3712323 0.85 CYP19A1 (0.46) CYP19A1CYP11B1CYP11B2XIAPBIRC2
SCHEMBL3711439 0.85 ADORA1 (0.46) CYP19A1CYP11B1CYP11B2XIAPBIRC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed