SCHEMBL3713586

SCHEMBL3713586

CCc1c(C=O)ccc(S(C)(=O)=O)c1F

nearest known ligand 0.32

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
ALDH1A1 P00352 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6851211 0.73 TDP1 (0.41) ALDH1A1L3MBTL1
SCHEMBL3714511 0.72 KAT6A (0.35) ALDH1A1
SCHEMBL2432111 0.71 ALDH1A1 (0.47) CYP2C9CYP2C19ALDH1A1L3MBTL1
SCHEMBL21358384 0.70 LMNA (0.36) ALDH1A1L3MBTL1
SCHEMBL28127127 0.69 ERN1 (0.38) CYP3A4CYP2C9CYP2C19ALDH1A1L3MBTL1
SCHEMBL3617240 0.69 ALDH3A1 (0.40) CYP3A4ALDH1A1
SCHEMBL28512785 0.68 L3MBTL1 (0.36) CYP3A4CYP2C9CYP2C19ALDH1A1L3MBTL1
SCHEMBL6076943 0.68 KDM4E (0.41) PTGS2ALDH1A1
SCHEMBL31005975 0.68 KDM4E (0.41) PTGS2ALDH1A1L3MBTL1
SCHEMBL2600012 0.68 KDM4E (0.41) PTGS2ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118208-A1 BENZOXAZEPIN-4- (5H) -YL DERIVATIVES AND THEIR USE TO TREAT CANCER EXELIXIS, INC. (US) 2010-10-14 WO disclosed