SCHEMBL3714749

SCHEMBL3714749

Cc1ccnc(CN2C=Cc3c(N)cccc3C2)c1-c1ccc(F)cc1Cl

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.33
HSD11B1 P28845 1/20 0.32
HTR1A P08908 1/20 0.32
HTR7 P34969 1/20 0.32
MAPK14 Q16539 3/20 0.31
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.31
CYP3A4 P08684 1/20 0.30
DPP4 P27487 1/20 0.30
DPP8 Q6V1X1 1/20 0.30
DPP9 Q86TI2 1/20 0.30
WDR5 P61964 1/20 0.30
MAPK13 O15264 1/20 0.30
MAPK12 P53778 1/20 0.30
MAPK11 Q15759 1/20 0.30
GRM2 Q14416 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3720425 0.83 FABP1 (0.37)
SCHEMBL21187438 0.67 HSD11B1 (0.42) HSD11B1MAPK14GRM2
SCHEMBL21187571 0.67 HSD11B1 (0.48) P2RX7HSD11B1HTR1AHTR7KDM4E
SCHEMBL7827660 0.66 PARP1 (0.35) POLBCYP3A4
SCHEMBL21187476 0.66 HSD11B1 (0.43) HSD11B1MAPK14
SCHEMBL3714746 0.62 DHFR (0.42) KDM4E
SCHEMBL21187496 0.61 NISCH (0.34) HSD11B1MAPK14
SCHEMBL21187487 0.61 TDO2 (0.35) HSD11B1MAPK14GRM2
SCHEMBL21187570 0.61 NISCH (0.42) HSD11B1MAPK14KDM4EPOLBDPP4
SCHEMBL27762859 0.60 PARP1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010117090-A1 NOVEL ISOQUINOLINYLOXYMETHYL HETEROARYL DERIVATIVES BANYU PHARMACEUTICAL CO.,LTD. (JP) 2010-10-14 WO claimed
WO-2010117090-A1 NOVEL ISOQUINOLINYLOXYMETHYL HETEROARYL DERIVATIVES BANYU PHARMACEUTICAL CO.,LTD. (JP) 2010-10-14 WO disclosed