SCHEMBL3717784

SCHEMBL3717784

NCc1cc(-c2ccc(Br)cc2)nc(NCCN2CCOCC2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 2/20 0.47
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
MKNK1 Q9BUB5 1/20 0.45
MAPK1 P28482 2/20 0.44
LMNA P02545 4/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
ACHE P22303 2/20 0.43
SCN9A Q15858 1/20 0.43
CYP3A4 P08684 2/20 0.42
BACE1 P56817 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CHRM1 P11229 1/20 0.42
CNR1 P21554 1/20 0.42
HTR2B P41595 1/20 0.42
KCNH2 Q12809 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3718051 0.86 ABL1 (0.49) ACP1KMT2AMEN1MKNK1LMNA
SCHEMBL3717779 0.82 SCN9A (0.58) ACP1KMT2AMEN1MKNK1MAPK1
SCHEMBL3722029 0.78 L3MBTL1 (0.44) KMT2AMEN1MAPK1LMNARAB9A
SCHEMBL3720912 0.76 MAPT (0.49) KMT2AMEN1MAPK1LMNANPC1
SCHEMBL3723261 0.76 PTGS1 (0.48) KMT2AMEN1MAPK1LMNANPC1
SCHEMBL3727322 0.72 AGTR1 (0.43) LMNAACHEALDH1A1
SCHEMBL3720119 0.71 ACP1 (0.44) ACP1LMNACYP1A2ALDH1A1
SCHEMBL13312433 0.71 ACP1 (0.61) ACP1KMT2AMEN1LMNANPC1
SCHEMBL3720305 0.70 PIK3CA (0.43) KMT2ACNR1
SCHEMBL3727142 0.70 AGTR1 (0.43) KMT2AMEN1LMNANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US disclosed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO disclosed