SCHEMBL3718259

SCHEMBL3718259

N#Cc1ncc(Oc2ccccc2C(F)(F)F)cc1F

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 3/20 0.43
AR P10275 14/20 0.43
LTA4H P09960 1/20 0.38
PTGS2 P35354 1/20 0.38
P2RY1 P47900 1/20 0.37
ERBB2 P04626 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3720603 0.80 MRGPRX1 (0.42) SLC22A12ARLTA4HPTGS2P2RY1
SCHEMBL3721302 0.79 AR (0.44) SLC22A12ARLTA4HPTGS2
SCHEMBL3718903 0.76 LTA4H (0.41) SLC22A12ARLTA4HPTGS2P2RY1
SCHEMBL3722454 0.75 P2RY1 (0.39) ARLTA4HPTGS2P2RY1
SCHEMBL3720604 0.74 P2RY1 (0.45) LTA4HPTGS2P2RY1
SCHEMBL1933633 0.73 AR (0.50) SLC22A12ARLTA4HPTGS2
SCHEMBL2132630 0.73 ALDH1A1 (0.40) AR
SCHEMBL3722554 0.73 P2RY1 (0.39) SLC22A12ARLTA4HPTGS2P2RY1
SCHEMBL8344932 0.72 HTR1A (0.47) SLC22A12ARP2RY1
SCHEMBL18615346 0.72 KMT2A (0.43) SLC22A12ARERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed