SCHEMBL3720604

SCHEMBL3720604

CC(=O)c1ncc(Oc2ccccc2C(F)(F)F)cc1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RY1 P47900 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
USP2 O75604 1/20 0.40
KMT2A Q03164 1/20 0.40
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
EGLN1 Q9GZT9 2/20 0.39
MRGPRX4 Q96LA9 1/20 0.38
NOTUM Q6P988 1/20 0.37
RXRA P19793 1/20 0.37
RXRB P28702 1/20 0.37
RXRG P48443 1/20 0.37
CDK8 P49336 1/20 0.37
LTA4H P09960 1/20 0.37
PTGS2 P35354 1/20 0.37
NFE2L2 Q16236 1/20 0.37
NR3C1 P04150 1/20 0.36
MRGPRX1 Q96LB2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3722554 0.85 P2RY1 (0.39) P2RY1SMN1; SMN2KDM4EMAPTUSP2
SCHEMBL3720603 0.80 MRGPRX1 (0.42) P2RY1LTA4HPTGS2MRGPRX1
SCHEMBL3722454 0.76 P2RY1 (0.39) P2RY1LTA4HPTGS2MRGPRX1
SCHEMBL3718259 0.74 SLC22A12 (0.43) P2RY1LTA4HPTGS2
SCHEMBL3718903 0.74 LTA4H (0.41) P2RY1MAOBMRGPRX4NOTUMCDK8
SCHEMBL2782296 0.72 PTGS2 (0.44) MAPTCDK8PTGS2
SCHEMBL11423116 0.71 P4HTM (0.50) MRGPRX4RXRARXRBRXRG
SCHEMBL11423110 0.70 KMT2A (0.50) SMN1; SMN2KMT2AMAOBLTA4HPTGS2
SCHEMBL14150163 0.69 LTA4H (0.45) P2RY1KDM4EKMT2ANOTUMRXRA
SCHEMBL30134107 0.69 KIF11 (0.38) SMN1; SMN2KDM4EMAPTUSP2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed