SCHEMBL3718665

SCHEMBL3718665

COc1cccc(CNc2nc(NCCCN)nc3c(C(C)C)n[nH]c23)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 3/20 0.44
ADORA2A P29274 4/20 0.42
ADORA2B P29275 4/20 0.42
ADORA1 P30542 4/20 0.42
ADORA3 P0DMS8 3/20 0.42
APP P05067 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
CCNE1 P24864 4/20 0.41
CDK2 P24941 4/20 0.41
CCNE2 O96020 2/20 0.41
CCNA2 P20248 2/20 0.41
CCNA1 P78396 2/20 0.41
STAT3 P40763 1/20 0.40
CCNB2 O95067 1/20 0.39
CCNB1 P14635 1/20 0.39
CCNB3 Q8WWL7 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
CDK5 Q00535 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3726417 0.88 TACR2 (0.42) CDK1APPCCNE1CDK2CCNE2
SCHEMBL3724956 0.88 CDK2 (0.42) CDK1APPCCNE1CDK2CCNE2
SCHEMBL2910733 0.87 CDK2 (0.52) CDK1APPCCNE1CDK2CCNE2
SCHEMBL3718660 0.84 CDK2 (0.55) CDK1CCNE1CDK2CCNE2CCNA2
SCHEMBL3714767 0.84 CDK2 (0.43) CDK1CCNE1CDK2CCNE2CCNA2
SCHEMBL3718378 0.82 CDK2 (0.43) CDK1MEN1KMT2ACCNE1CDK2
SCHEMBL3720176 0.82 TACR2 (0.49) CDK1CCNE1CDK2CCNE2CCNA2
SCHEMBL3725653 0.82 CDK2 (0.46) CDK1CCNE1CDK2CCNE2CCNA2
SCHEMBL3799897 0.81 CDK2 (0.56) CDK1CCNE1CDK2CCNE2CCNA2
SCHEMBL2910995 0.81 CDK2 (0.52) CDK1APPCCNE1CDK2CCNE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010139288-A1 5,7-DISUBSTITUTED 3-ISOPROPYLPYRAZOLO[4,3-D]PYRIMIDINES FOR USE AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS C3 BIO GMBH (DE) 2010-12-09 WO disclosed