SCHEMBL3726417

SCHEMBL3726417

CC(C)c1n[nH]c2c(NCc3cccc(Cl)c3)nc(NCCCN)nc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 1/20 0.42
CDK2 P24941 5/20 0.42
CCNE1 P24864 4/20 0.42
CCNE2 O96020 2/20 0.42
CCNA2 P20248 2/20 0.42
CCNA1 P78396 2/20 0.42
CDK9 P50750 1/20 0.42
TMIGD3 P0DMS9 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
GRM4 Q14833 1/20 0.40
PLK4 O00444 1/20 0.40
PAK4 O96013 1/20 0.40
CDK1 P06493 2/20 0.40
CCNB2 O95067 1/20 0.40
CCNB1 P14635 1/20 0.40
CCNB3 Q8WWL7 1/20 0.40
PDE2A O00408 1/20 0.39
CDK5 Q00535 2/20 0.39
APP P05067 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3724956 0.89 CDK2 (0.42) TACR2CDK2CCNE1CCNE2CCNA2
SCHEMBL3720176 0.88 TACR2 (0.49) TACR2CDK2CCNE1CCNE2CCNA2
SCHEMBL2910733 0.88 CDK2 (0.52) TACR2CDK2CCNE1CCNE2CCNA2
SCHEMBL3718665 0.88 CDK1 (0.44) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL3714767 0.87 CDK2 (0.43) TACR2CDK2CCNE1CCNE2CCNA2
SCHEMBL3724487 0.84 CDK2 (0.47) TACR2CDK2CCNE1CCNE2CCNA2
SCHEMBL3719064 0.84 CYP3A4 (0.43) TACR2CDK2CCNE1CCNE2CCNA2
SCHEMBL3726416 0.84 CDK2 (0.56) CDK2CCNE1CCNE2CCNA2CDK9
SCHEMBL3725653 0.82 CDK2 (0.46) TACR2CDK2CCNE1CCNE2CCNA2
SCHEMBL2910995 0.82 CDK2 (0.52) CDK2CCNE1CCNE2CCNA2CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010139288-A1 5,7-DISUBSTITUTED 3-ISOPROPYLPYRAZOLO[4,3-D]PYRIMIDINES FOR USE AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS C3 BIO GMBH (DE) 2010-12-09 WO disclosed