SCHEMBL3725653

SCHEMBL3725653

CC(C)c1n[nH]c2c(NCc3ccc(F)cc3)nc(NCCCN)nc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 8/20 0.46
CCNE1 P24864 7/20 0.46
CCNE2 O96020 3/20 0.46
CCNA2 P20248 3/20 0.46
CCNA1 P78396 3/20 0.46
CDK5 Q00535 4/20 0.43
STK17A Q9UEE5 2/20 0.39
TACR2 P21452 1/20 0.39
CCNB2 O95067 2/20 0.38
CDK1 P06493 2/20 0.38
CCNB1 P14635 2/20 0.38
CCNB3 Q8WWL7 2/20 0.38
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
STK17B O94768 1/20 0.37
CTNNB1 P35222 1/20 0.37
TCF7L2 Q9NQB0 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
PLK4 O00444 1/20 0.36
PAK4 O96013 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3714767 0.90 CDK2 (0.43) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL3720176 0.90 TACR2 (0.49) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL2910733 0.90 CDK2 (0.52) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL3724956 0.88 CDK2 (0.42) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL3716187 0.86 CDK2 (0.43) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL3718696 0.86 CDK2 (0.43) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL3721963 0.85 P2RX7 (0.41) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL3724809 0.84 CDK2 (0.40) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL2910995 0.83 CDK2 (0.52) CDK2CCNE1CCNE2CCNA2CCNA1
SCHEMBL3725652 0.82 CDK2 (0.62) CDK2CCNE1CCNE2CCNA2CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010139288-A1 5,7-DISUBSTITUTED 3-ISOPROPYLPYRAZOLO[4,3-D]PYRIMIDINES FOR USE AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS C3 BIO GMBH (DE) 2010-12-09 WO disclosed