SCHEMBL3718985

SCHEMBL3718985

COc1ccc(Oc2ccc(CN)nc2)c(Br)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 2/20 0.39
MEN1 O00255 2/20 0.39
MAPT P10636 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 2/20 0.39
TAAR1 Q96RJ0 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
P2RX3 P56373 1/20 0.38
P2RX2 Q9UBL9 1/20 0.38
ADRA2A P08913 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
ALDH1A1 P00352 1/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3721624 0.84 MPO (0.44) ADRA1AMEN1KMT2ATAAR1P2RX3
SCHEMBL3722011 0.82 ADRA1A (0.43) ADRA1AMEN1MAPTKMT2ATAAR1
SCHEMBL3726016 0.81 L3MBTL1 (0.40) ADRA1AMAPTTAAR1NPSR1HTR2A
SCHEMBL10002478 0.79 MAOB (0.43) TAAR1CA12CA1CA2CA7
SCHEMBL3725866 0.79 P2RX3 (0.40) ADRA1AMEN1MAPTKMT2AKDM4E
SCHEMBL3721554 0.79 TAAR1 (0.38) ADRA1AMEN1MAPTKMT2AKDM4E
Hydrochloric Acid SCHEMBL3722878 0.78 MEN1 (0.40) ADRA1AMEN1MAPTKMT2AKDM4E
Hydrochloric Acid SCHEMBL20447729 0.78 MAOB (0.46) TAAR1CA12CA1CA2CA7
SCHEMBL12239019 0.77 ST14 (0.52) ADRA1AMEN1MAPTKMT2AKDM4E
SCHEMBL16853366 0.76 ST14 (0.40) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed