SCHEMBL3722011

SCHEMBL3722011

COc1ccc(Oc2ccc(CN)nc2)c(C(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 4/20 0.43
ADRA2A P08913 2/20 0.43
P2RX3 P56373 2/20 0.43
P2RX2 Q9UBL9 2/20 0.43
CYP2D6 P10635 2/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPK1 P28482 1/20 0.39
BLM P54132 1/20 0.39
TAAR1 Q96RJ0 1/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
HTR2A P28223 1/20 0.35
ADRB2 P07550 1/20 0.34
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
CA1 P00915 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3718985 0.82 ADRA1A (0.39) ADRA1AADRA2AP2RX3P2RX2MEN1
SCHEMBL3721624 0.81 MPO (0.44) ADRA1AADRA2AP2RX3P2RX2MEN1
SCHEMBL3726016 0.81 L3MBTL1 (0.40) ADRA1ATAAR1LMNAHTR2AMAPT
SCHEMBL3726572 0.79 NQO1 (0.43) ADRA1AADRA2AP2RX3P2RX2CYP2D6
SCHEMBL10002478 0.76 MAOB (0.43) MAPK1TAAR1CA1CA2ALDH1A1
Hydrochloric Acid SCHEMBL20447729 0.75 MAOB (0.46) MAPK1TAAR1CA1CA2ALDH1A1
SCHEMBL16148146 0.73 CYP2D6 (0.59) ADRA1AADRA2ACYP2D6MEN1KMT2A
SCHEMBL16853366 0.73 ST14 (0.40) TSHRALDH1A1
SCHEMBL3730285 0.69 NR3C1 (0.34) LMNAHTR2AMAPT
SCHEMBL19555693 0.69 MBOAT4 (0.45) MAPK1RXRAGRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed