SCHEMBL3720102

SCHEMBL3720102

COc1ccc(Oc2ccc3nc(CCN)ccc3c2)c(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 3/20 0.47
NCF1 P14598 1/20 0.45
TAAR1 Q96RJ0 2/20 0.42
ADRA1A P35348 1/20 0.42
SLC6A4 P31645 4/20 0.40
HTR2A P28223 3/20 0.40
NQO1 P15559 1/20 0.40
SLC6A2 P23975 1/20 0.39
SLC6A3 Q01959 1/20 0.39
CHEK2 O96017 1/20 0.39
ALDH1A1 P00352 2/20 0.38
GFER P55789 1/20 0.38
KCNH2 Q12809 2/20 0.38
DYRK1A Q13627 1/20 0.38
KDM4E B2RXH2 1/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
HDAC1 Q13547 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14352239 0.86 NCF1 (0.58) PDE10ANCF1TAAR1ADRA1ANQO1
SCHEMBL3726423 0.82 MTNR1A (0.47) PDE10A
SCHEMBL3717395 0.82 HDAC1 (0.42) PDE10ANCF1SLC6A4HTR2ANQO1
SCHEMBL3717394 0.77 HDAC8 (0.44) NCF1NQO1CHEK2ALDH1A1KCNH2
SCHEMBL5928217 0.77 NCF1 (0.54) PDE10ANCF1TAAR1ADRA1ANQO1
SCHEMBL3720101 0.76 HTR1A (0.44) PDE10ANCF1SLC6A4HTR2ANQO1
SCHEMBL28254830 0.74 NCF1 (0.62) PDE10ANCF1NQO1ALDH1A1GFER
SCHEMBL14127808 0.73 NCF1 (0.56) PDE10ANCF1NQO1SLC6A2SLC6A3
SCHEMBL27596905 0.72 NCF1 (0.54) PDE10ANCF1NQO1SLC6A2SLC6A3
SCHEMBL3721624 0.72 MPO (0.44) TAAR1ADRA1ASLC6A4HTR2ASLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed