SCHEMBL3720159

SCHEMBL3720159

CC(=O)c1ccc2nc(Oc3ccc(SC(C)C)c(C)c3C)ccc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.42
CYP2A6 P11509 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
ALDH1A1 P00352 6/20 0.33
MAPK1 P28482 1/20 0.33
KMT2A Q03164 2/20 0.32
GAA P10253 1/20 0.32
MEN1 O00255 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
SCN7A Q01118 1/20 0.31
KCNH2 Q12809 1/20 0.31
SCN9A Q15858 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HDAC9 Q9UKV0 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3717722 0.84 PDE4B (0.45) PDE4BCYP2A6SMN1; SMN2ALDH1A1KMT2A
SCHEMBL3720271 0.83 PDE4B (0.42) PDE4BCYP2A6SMN1; SMN2ALDH1A1MAPK1
SCHEMBL3720626 0.83 ACACB (0.37)
SCHEMBL3720627 0.81 MTNR1A (0.50) SMN1; SMN2ALDH1A1SCN9AHPGDMAPT
SCHEMBL3720536 0.80 PDE4B (0.42) PDE4BCYP2A6SMN1; SMN2ALDH1A1MAPK1
SCHEMBL3719889 0.80 PDE4B (0.42) PDE4BCYP2A6SMN1; SMN2ALDH1A1MAPK1
SCHEMBL3720162 0.80 ALDH1A1 (0.31) SMN1; SMN2ALDH1A1HPGDHTT
SCHEMBL3727136 0.77 MAPT (0.34) MAPT
SCHEMBL3727138 0.77 TSHR (0.34) SMN1; SMN2MAPK1KMT2AMEN1TSHR
SCHEMBL3720632 0.77 PDE4B (0.53) PDE4BCYP2A6SMN1; SMN2ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed