SCHEMBL3720271

SCHEMBL3720271

CC(=O)c1ccc2nc(Oc3ccc(SC(C)C)cc3C)ccc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
HIF1A Q16665 1/20 0.36
MAPK14 Q16539 2/20 0.35
ALDH1A1 P00352 6/20 0.35
MAPK1 P28482 1/20 0.35
CYP2A6 P11509 1/20 0.35
PPARG P37231 1/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ABL1 P00519 1/20 0.32
GAA P10253 1/20 0.32
SCN7A Q01118 1/20 0.31
KCNH2 Q12809 1/20 0.31
SCN9A Q15858 1/20 0.31
HDAC3 O15379 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3719889 0.88 PDE4B (0.42) PDE4BSMN1; SMN2LMNACYP1A2CYP2C19
SCHEMBL3720536 0.88 PDE4B (0.42) PDE4BSMN1; SMN2LMNACYP1A2CYP2C19
SCHEMBL3717153 0.86 PDE4B (0.43) PDE4BSMN1; SMN2LMNAMAPK14ALDH1A1
SCHEMBL3720632 0.84 PDE4B (0.53) PDE4BSMN1; SMN2LMNACYP1A2CYP2C19
SCHEMBL3720159 0.83 PDE4B (0.42) PDE4BSMN1; SMN2ALDH1A1MAPK1CYP2A6
SCHEMBL3717454 0.83 ACACB (0.37) SMN1; SMN2LMNACYP1A2CYP2C19HIF1A
SCHEMBL3721868 0.82 PDE4B (0.48) PDE4BMAPK14ALDH1A1CYP2A6KMT2A
SCHEMBL3717633 0.82 PDE4B (0.47) PDE4BSMN1; SMN2CYP1A2CYP2C19MAPK14
SCHEMBL3717456 0.81 MTNR1A (0.50) SMN1; SMN2LMNACYP1A2CYP2C19HIF1A
SCHEMBL3720275 0.80 LMNA (0.32) SMN1; SMN2LMNACYP1A2CYP2C19HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed