SCHEMBL3721091

SCHEMBL3721091

NCc1cc(-c2ccc3c(c2)OCO3)nc(N2CCN(Cc3ccc4c(c3)OCO4)CC2)n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
CYP1A2 P05177 2/20 0.57
CYP3A4 P08684 2/20 0.57
CYP2D6 P10635 2/20 0.57
CYP2C19 P33261 2/20 0.57
USP2 O75604 1/20 0.57
HTR1A P08908 1/20 0.57
ADRA2A P08913 1/20 0.57
DRD2 P14416 1/20 0.57
ADRA2B P18089 1/20 0.57
ADRA2C P18825 1/20 0.57
NFKB1 P19838 1/20 0.57
SLC6A2 P23975 1/20 0.57
MAPK1 P28482 1/20 0.57
SLC6A4 P31645 1/20 0.57
ADRA1A P35348 1/20 0.57
DRD3 P35462 1/20 0.57
HTR2B P41595 1/20 0.57
KCNH2 Q12809 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3720812 0.90 LMNA (0.59) MEN1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL3724689 0.84 MEN1 (0.50) MEN1KMT2ACYP1A2CYP3A4CYP2C19
SCHEMBL3728043 0.81 ADORA1 (0.44) NFKB1MAPK1HSD17B10POLBLMNA
SCHEMBL3725556 0.80 ABCB1 (0.56) NFKB1HSD17B10LMNAKDM4EALDH1A1
SCHEMBL3718806 0.80 KDM4E (0.49) MEN1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL3719736 0.76 NPC1 (0.45) MEN1KMT2AUSP2NFKB1SLC6A2
SCHEMBL3720809 0.74 LMNA (0.54) MEN1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL108678 0.74 KDM4E (0.70) MEN1KMT2ACYP1A2CYP3A4CYP2D6
Piribedil SCHEMBL29359749 0.74 MEN1 (1.00) MEN1KMT2ACYP1A2CYP3A4CYP2D6
Piribedil SCHEMBL5605887 0.74 MEN1 (1.00) MEN1KMT2ACYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO disclosed