SCHEMBL3721099

SCHEMBL3721099

NCc1cc(-c2ccccc2F)nc(N2CCN(c3ccccc3F)CC2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.44
ALDH1A1 P00352 5/20 0.44
LMNA P02545 3/20 0.44
NPC1 O15118 1/20 0.44
AGER Q15109 1/20 0.42
TSHR P16473 2/20 0.40
KDM4E B2RXH2 2/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 2/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HSD17B10 Q99714 1/20 0.39
DRD4 P21917 2/20 0.39
DRD3 P35462 1/20 0.39
USP2 O75604 1/20 0.39
MAPK1 P28482 1/20 0.39
ABCB1 P08183 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3724503 0.91 CYP11B2 (0.46) SMN1; SMN2ALDH1A1LMNANPC1AGER
SCHEMBL3726395 0.91 LMNA (0.41) SMN1; SMN2ALDH1A1LMNANPC1AGER
SCHEMBL3717799 0.91 SMN1; SMN2 (0.41) SMN1; SMN2ALDH1A1LMNANPC1AGER
SCHEMBL3718590 0.88 ALDH1A1 (0.52) SMN1; SMN2ALDH1A1LMNANPC1TSHR
SCHEMBL3721047 0.86 SMN1; SMN2 (0.45) SMN1; SMN2ALDH1A1LMNANPC1TSHR
SCHEMBL3727042 0.86 DRD2 (0.47) SMN1; SMN2ALDH1A1LMNANPC1TSHR
SCHEMBL3721920 0.86 LMNA (0.52) SMN1; SMN2ALDH1A1LMNANPC1MAPT
SCHEMBL3720203 0.86 KMT2A (0.42) SMN1; SMN2ALDH1A1LMNANPC1AGER
SCHEMBL3720273 0.85 ALDH1A1 (0.44) SMN1; SMN2ALDH1A1LMNANPC1TSHR
SCHEMBL3721161 0.84 MAPT (0.44) SMN1; SMN2ALDH1A1LMNANPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US claimed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO claimed
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US disclosed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO disclosed