SCHEMBL3721164

SCHEMBL3721164

Nc1nc(C(=O)O)cc(-c2ccc(C#Cc3ccc(CN4CCOCC4)cc3)cc2)n1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.47
JAK2 O60674 1/20 0.46
HRH3 Q9Y5N1 1/20 0.44
BCHE P06276 1/20 0.44
MAOA P21397 1/20 0.44
ACHE P22303 1/20 0.44
MAOB P27338 1/20 0.44
MMP2 P08253 1/20 0.44
MMP8 P22894 1/20 0.44
MMP13 P45452 1/20 0.44
MOK Q9UQ07 1/20 0.43
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3716618 0.89 MMP2 (0.48) MMP2MMP8MMP13
SCHEMBL3715918 0.88 MAPK1 (0.45) PARP1JAK2BCHEMAOAACHE
SCHEMBL3709302 0.84 BCHE (0.44) PARP1JAK2BCHEMAOAACHE
SCHEMBL3709560 0.83 KMO (0.50) HRH3BCHEMAOAACHEMAOB
SCHEMBL3715177 0.81 TLR7 (0.44) MOK
SCHEMBL3709419 0.80 PARP1 (0.45) PARP1HRH3MMP2MMP8MMP13
SCHEMBL13188620 0.79 KMO (0.47) HRH3BCHEMAOAACHEMAOB
SCHEMBL3714253 0.77 HDAC1 (0.52) MMP2MMP8MMP13
SCHEMBL3713943 0.77 MAPK1 (0.45) MMP2MMP8MMP13
SCHEMBL3712370 0.77 ACP1 (0.47) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed