SCHEMBL3722003

SCHEMBL3722003

COc1ccc(Oc2cnc(C#N)nc2)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 6/20 0.46
SLC6A4 P31645 4/20 0.45
SLC6A2 P23975 1/20 0.45
SLC6A3 Q01959 1/20 0.45
HTR2A P28223 3/20 0.43
HPGDS O60760 1/20 0.40
KCNH2 Q12809 2/20 0.40
DYRK1A Q13627 1/20 0.40
ABL1 P00519 1/20 0.40
BCR P11274 1/20 0.40
SRC P12931 1/20 0.40
MPO P05164 1/20 0.39
TPO P07202 1/20 0.39
EPX P11678 1/20 0.39
LPO P22079 1/20 0.39
AR P10275 2/20 0.39
HPGD P15428 1/20 0.39
POLB P06746 1/20 0.38
GAA P10253 1/20 0.38
S1PR4 O95977 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3719152 0.80 AR (0.48) SLC22A12AR
SCHEMBL2788214 0.79 AR (0.55) SLC6A4SLC6A2SLC6A3HTR2AKCNH2
SCHEMBL756234 0.78 AR (0.62) SLC22A12SLC6A4SLC6A2SLC6A3HTR2A
SCHEMBL3721298 0.77 SLC6A4 (0.45) SLC6A4SLC6A2SLC6A3HTR2AKCNH2
SCHEMBL16507366 0.74 ALDH1A1 (0.53) SLC22A12SLC6A4SLC6A2SLC6A3HPGDS
SCHEMBL16175273 0.74 SLC22A12 (0.49) SLC22A12SLC6A4SLC6A3HTR2AKCNH2
SCHEMBL2185557 0.74 NAAA (0.42) HPGDSSRCPOLBGAA
SCHEMBL3725814 0.73 SLC6A4 (0.44) SLC22A12SLC6A4SLC6A2SLC6A3HTR2A
SCHEMBL3721624 0.73 MPO (0.44) SLC22A12SLC6A4SLC6A2SLC6A3HTR2A
SCHEMBL15832086 0.73 POLB (0.47) SLC22A12ABL1BCRSRCPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed