SCHEMBL3724725

SCHEMBL3724725

Nc1cc(CN2CCNC(=O)C2)cc2cc(-c3cccc(F)c3)n(C3CCCC3)c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
HTR6 P50406 1/20 0.39
ALK Q9UM73 1/20 0.39
GRM2 Q14416 1/20 0.38
CDK4 P11802 1/20 0.38
CDK6 Q00534 1/20 0.38
MCHR1 Q99705 2/20 0.37
EGFR P00533 1/20 0.36
ERBB2 P04626 1/20 0.36
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
CYP11B2 P19099 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
OGFRL1 Q5TC84 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3729429 0.83 JAK2 (0.40) JAK2JAK1ALKGRM2CDK4
SCHEMBL3015318 0.72 VCP (0.42) JAK2JAK1HTR6ALKGRM2
SCHEMBL31043038 0.72 VCP (0.42) JAK2JAK1HTR6ALKGRM2
SCHEMBL3758694 0.70 JAK1 (0.39) JAK2JAK1OPRM1OPRD1OPRK1
SCHEMBL17554234 0.64 JAK1 (0.39) JAK2JAK1KMT2AMEN1OPRM1
SCHEMBL4748942 0.64 ALDH1A1 (0.61) GRM2MCHR1KMT2AMEN1ALDH1A1
SCHEMBL3015320 0.62 BTK (0.37) JAK2JAK1HTR6ALKGRM2
SCHEMBL3149433 0.62 ALDH1A1 (0.50) JAK2JAK1GRM2KMT2AMEN1
SCHEMBL220097 0.61 SIGMAR1 (0.62) KMT2AMEN1ALDH1A1
SCHEMBL3038501 0.61 SMN1; SMN2 (0.56) KMT2AMEN1CYP11B2ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2178870-A1 INDOLE AND INDAZOLE COMPOUNDS AS AN INHIBITOR OF CELLULAR NECROSIS LG Life Sciences Ltd. (KR) 2010-04-28 EP claimed
WO-2009025478-A1 INDOLE AND INDAZOLE COMPOUNDS AS AN INHIBITOR OF CELLULAR NECROSIS LG LIFE SCIENCES LTD. (KR) 2009-02-26 WO claimed
EP-2178870-A1 INDOLE AND INDAZOLE COMPOUNDS AS AN INHIBITOR OF CELLULAR NECROSIS LG Life Sciences Ltd. (KR) 2010-04-28 EP disclosed
WO-2009025478-A1 INDOLE AND INDAZOLE COMPOUNDS AS AN INHIBITOR OF CELLULAR NECROSIS LG LIFE SCIENCES LTD. (KR) 2009-02-26 WO disclosed