SCHEMBL3724487

SCHEMBL3724487

CC(C)c1n[nH]c2c(NCc3cc(Cl)ccc3O)nc(NCCCN)nc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 11/20 0.47
CCNE1 P24864 10/20 0.47
CDK9 P50750 6/20 0.47
CCNT1 O60563 5/20 0.47
CCNE2 O96020 3/20 0.47
CCNT2 O60583 1/20 0.47
CDK5 Q00535 5/20 0.44
CDK5R1 Q15078 5/20 0.44
CDK7 P50613 4/20 0.44
CCNH P51946 4/20 0.44
TACR2 P21452 1/20 0.42
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
MAPT P10636 2/20 0.39
HTT P42858 2/20 0.39
CHEK1 O14757 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
CDK1 P06493 2/20 0.37
CCNB2 O95067 1/20 0.37
CCNB1 P14635 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3718696 0.89 CDK2 (0.43) CDK2CCNE1CDK9CCNT1CCNE2
SCHEMBL3720176 0.86 TACR2 (0.49) CDK2CCNE1CCNE2CDK5CDK5R1
SCHEMBL3724482 0.85 CDK2 (0.51) CDK2CCNE1CDK9CCNT1CCNE2
SCHEMBL3726417 0.84 TACR2 (0.42) CDK2CCNE1CDK9CCNE2CDK5
SCHEMBL3719064 0.83 CYP3A4 (0.43) CDK2CCNE1CCNE2CDK5TACR2
SCHEMBL3721963 0.81 P2RX7 (0.41) CDK2CCNE1CCNE2CDK5TACR2
SCHEMBL3714767 0.81 CDK2 (0.43) CDK2CCNE1CCNE2CDK5TACR2
SCHEMBL3719455 0.81 CDK2 (0.52) CDK2CCNE1CDK9CCNT1CCNE2
SCHEMBL3716187 0.81 CDK2 (0.43) CDK2CCNE1CCNE2CDK5CDK5R1
SCHEMBL2910733 0.80 CDK2 (0.52) CDK2CCNE1CDK9CCNT1CCNE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010139288-A1 5,7-DISUBSTITUTED 3-ISOPROPYLPYRAZOLO[4,3-D]PYRIMIDINES FOR USE AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS C3 BIO GMBH (DE) 2010-12-09 WO disclosed