SCHEMBL3727460

SCHEMBL3727460

CSc1nc(Cl)c2ncn(COC(=O)C(C)(C)C)c2n1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 12/20 0.38
HSP90AA1 P07900 11/20 0.38
P2RX7 Q99572 2/20 0.36
ABCB11 O95342 1/20 0.36
POLA1 P09884 1/20 0.36
POLG P54098 1/20 0.36
FAP Q12884 1/20 0.36
SLC22A6 Q4U2R8 1/20 0.36
HDAC6 Q9UBN7 5/20 0.35
HDAC1 Q13547 4/20 0.35
HDAC4 P56524 1/20 0.35
HSP90B1 P14625 1/20 0.33
TRAP1 Q12931 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20774171 0.85 P2RX7 (0.49) HSP90AB1HSP90AA1P2RX7ABCB11POLA1
SCHEMBL3730211 0.84 HSP90AB1 (0.49) HSP90AB1HSP90AA1HDAC6HDAC1HDAC4
SCHEMBL21282838 0.76 CDK1 (0.46) HSP90AB1HSP90AA1P2RX7
SCHEMBL31599667 0.71 FGFR1 (0.41) ABCB11POLA1POLGFAPSLC22A6
SCHEMBL7672450 0.71 PNP (0.63)
SCHEMBL10364108 0.70 ACHE (0.40) HDAC6HDAC1HDAC4
SCHEMBL11082532 0.68 ABCB11 (0.45) ABCB11POLA1POLGFAPSLC22A6
SCHEMBL21282810 0.68 CDK1 (0.47) HSP90AB1HSP90AA1
SCHEMBL2780215 0.68 PNP (0.43)
SCHEMBL16510025 0.67 POLB (0.42) ABCB11POLA1POLGFAPSLC22A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7825126-B2 Purine derivatives as A3 and A1 adenosine receptor agonists THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2010-11-02 US disclosed
US-20070232626-A1 Purine Derivatives as A3 and A1 Adenosine Receptor Agonists GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPT OF HEALTH AND H (MD) 2007-10-04 US disclosed
EP-1794162-A1 PURINE DERIVATIVES AS A3 AND A1 ADENOSINE RECEPTOR AGONISTS The Government of the United States of America, as repres. by the Secretary of Health and Human Services, Nat. Inst. of Health (US) 2007-06-13 EP disclosed
WO-2006031505-A1 PURINE DERIVATIVES AS A3 AND A1 ADENOSINE RECEPTOR AGONISTS GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2006-03-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070232626-A1 Purine Derivatives as A3 and A1 Adenosine Receptor Agonists ADORA1, ADORA3, ADORA2A HSP90AB1 3062/4885HSP90AA1 2331/4885P2RX7 9/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.