SCHEMBL374641

SCHEMBL374641

O=C(O)c1ccccc1Nc1c(Cl)cccc1Cl

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FTO Q9C0B1 10/20 0.71
PBRM1 Q86U86 1/20 0.71
CLCN2 P51788 7/20 0.70
MEN1 O00255 2/20 0.69
TTR P02766 2/20 0.69
ADORA3 P0DMS8 2/20 0.69
PTGS2 P35354 2/20 0.69
AKR1C3 P42330 2/20 0.69
KMT2A Q03164 2/20 0.69
USP2 O75604 1/20 0.69
MT-CO2 P00403 1/20 0.69
LMNA P02545 1/20 0.69
PLA2G1B P04054 1/20 0.69
CYP1A2 P05177 1/20 0.69
PGR P06401 1/20 0.69
CYP3A4 P08684 1/20 0.69
HTR1A P08908 1/20 0.69
ADRA2A P08913 1/20 0.69
AR P10275 1/20 0.69
MAPT P10636 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3500411 0.89 FTO (0.72) FTOPBRM1CLCN2MEN1TTR
SCHEMBL24021600 0.86 FTO (0.77) FTOCLCN2TTR
SCHEMBL11518282 0.86 PTGS2 (0.56) FTOPBRM1CLCN2MEN1TTR
SCHEMBL374772 0.86 PTGS2 (0.55) FTOPBRM1CLCN2MEN1TTR
SCHEMBL4249088 0.85 PBRM1 (0.75) FTOPBRM1CLCN2MEN1TTR
SCHEMBL30575470 0.85 PBRM1 (0.75) FTOPBRM1CLCN2MEN1TTR
SCHEMBL11407549 0.84 CXCL8 (0.55) FTOPBRM1CLCN2MEN1TTR
Clofenamic Acid SCHEMBL1477650 0.84 PBRM1 (0.73) FTOPBRM1CLCN2MEN1TTR
Clofenamic Acid SCHEMBL29900200 0.84 PBRM1 (0.73) FTOPBRM1CLCN2MEN1TTR
SCHEMBL28297347 0.84 PBRM1 (0.73) FTOPBRM1CLCN2MEN1TTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 49 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108047068-A A kind of synthetic method of C14H10Cl2NNaO2 impurity B 河南中帅医药科技股份有限公司 2018-05-18 CN claimed
JP-55108845-A None JP disclosed
JP-56079651-A None JP disclosed
CN-111808011-B High penetration composition and its application 泰飞尔生物医药(苏州)有限公司 2024-02-27 CN disclosed
CN-109553544-B Method for synthesizing diclofenac sodium 浙江普利药业有限公司 2022-02-08 CN disclosed
US-11173137-B2 Compositions and methods to modulate chloride ion channel activity THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2021-11-16 US disclosed
CN-102164594-B Use of anti-connexin agents for modulating the efficacy of psychotropic drug molecules 原子能和替代能源委员会 2021-09-28 CN disclosed
CN-113402408-A Method for synthesizing diclofenac sodium 河南康达制药有限公司 2021-09-17 CN disclosed
WO-2020037294-A1 SYSTEM AND METHOD FOR BIPHASIC TRANSDERMAL IONTOPHORETIC DELIVERY OF DICLOPHENAC AND OTHER THERAPEUTIC AGENTS INCUBE LABS, LLC (US) 2020-02-20 WO disclosed
CN-109553544-A A kind of synthetic method of C14H10Cl2NNaO2 浙江普利药业有限公司 2019-04-02 CN disclosed
US-5112846-A Nonsteroidal antiinflammatory agents WARNER-LAMBERT COMPANY (US) 1992-05-12 US disclosed
US-5075330-A N-hydroxyamide, N-hydroxythioamide, N-hydroxyurea, and N-hydroxythiourea derivatives of selected NSAIDS as antiinflammatory agents WARNER-LAMBERT CO. (US) 1991-12-24 US disclosed
US-4981865-A N-hydroxyamide, N-hydroxythioamide, hydroxyurea, and N-hydroxythiourea derivatives of selected nsaids as antiinflammatory agents WARNER-LAMBERT CO. (US) 1991-01-01 US disclosed
EP-0316630-A1 Novel fenamic acid hydroxamate derivatives having cyclooxygenase and 5-lipoxygenase inhibition WARNER-LAMBERT COMPANY (US) 1989-05-24 EP disclosed
WO-1989003818-A1 NOVEL FENAMIC ACID HYDROXAMATE DERIVATIVES HAVING CYCLOOXYGENASE AND 5-LIPOXYGENASE INHIBITION WARNER-LAMBERT COMPANY (US) 1989-05-05 WO disclosed
JP-S5679651-A PREPARATION OF BENZALDEHYDE DERIVATIVE PAAMAKEMU ASIA:KK 1981-06-30 JP disclosed
US-4242522-A O-(N-Allyl-2,6-dichloroanilino)phenylacetic acid derivative and a process for preparing the same NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1980-12-30 US disclosed
JP-S55108845-A PREPARATION OF SUBSTITUTED PHENYLACETIC ACID DERIVATIVE PAAMAKEMU ASIA:KK 1980-08-21 JP disclosed
US-4189595-A [N-benzyl-o-(2,6-dichloroanilino)phenyl]acetic acid derivatives NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1980-02-19 US disclosed
US-4188343-A Process for preparing anthranylaldehyde derivatives NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1980-02-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11173137-B2 Compositions and methods to modulate chloride ion channel activity CLCN2, CLIC1, CLIC4 FTO 4582/4885PBRM1 3615/4885CLCN2 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.