SCHEMBL3752171

SCHEMBL3752171

Cc1nc(-c2ccc(C(F)(F)F)cc2)sc1C(OCC(F)(F)C1CC1)c1ccc(-c2noc(=O)[nH]2)cc1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 3/20 0.37
PPARD Q03181 2/20 0.37
MDM2 Q00987 1/20 0.37
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
FFAR1 O14842 9/20 0.35
BPGM P07738 1/20 0.35
CHRM5 P08912 1/20 0.35
SLC6A3 Q01959 1/20 0.35
PLA2G2A P14555 4/20 0.34
PLA2G10 O15496 2/20 0.34
PLA2G1B P04054 2/20 0.34
PLA2G5 P39877 2/20 0.34
RARB P10826 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3744980 0.88 ALDH1A1 (0.38) PPARAPPARDMDM2NPC1ALDH1A1
SCHEMBL3748585 0.86 BPGM (0.37) PPARAPPARDNPC1ALDH1A1GAA
SCHEMBL3747892 0.86 PLA2G2A (0.42) PPARAPPARDNPC1ALDH1A1GAA
SCHEMBL3745605 0.82 PLAT (0.36) PPARAPPARDMDM2NPC1ALDH1A1
SCHEMBL3752165 0.82 PPARD (0.37) PPARAPPARDMDM2NPC1ALDH1A1
SCHEMBL3743853 0.81 NPC1 (0.36) PPARAPPARDNPC1ALDH1A1GAA
SCHEMBL3753667 0.80 PPARD (0.36) PPARAPPARDMDM2NPC1ALDH1A1
SCHEMBL3527489 0.80 BPGM (0.38) MDM2ALDH1A1BPGMPLA2G2APLA2G10
SCHEMBL3525623 0.77 ALDH1A1 (0.37) ALDH1A1BPGMPLA2G2APLA2G10PLA2G1B
SCHEMBL3747886 0.77 PPARD (0.40) PPARAPPARDNPC1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1931660-B1 PHENYL-[1,2,4]-OXADIAZOL-5-ONE DERIVATIVES WITH PHENYL GROUP, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS SANOFI SA (FR) 2012-08-01 EP claimed
EP-1931660-B1 PHENYL-[1,2,4]-OXADIAZOL-5-ONE DERIVATIVES WITH PHENYL GROUP, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS SANOFI SA (FR) 2012-08-01 EP disclosed
US-7834030-B2 Phenyl-[1,2,4]-oxadiazol-5-one derivatives, pharmaceutical compositions and therapeutic use thereof SANOFI-AVENTIS (FR) 2010-11-16 US disclosed
US-20080262036-A1 Phenyl-[1,2,4]-oxadiazol-5-one Derivatives, Pharmaceutical Compositions and Therapeutic Use Thereof SANOFI-AVENTIS (FR) 2008-10-23 US disclosed
EP-1931660-A2 PHENYL-[1,2,4]-OXADIAZOL-5-ONE DERIVATIVES WITH PHENYL GROUP, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS Sanofi-Aventis (FR) 2008-06-18 EP disclosed
WO-2007039178-A2 PHENYL-[1,2,4]-OXADIAZOL-5-ONE DERIVATIVES WITH PHENYL GROUP, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS SANOFI-AVENTIS (DE) 2007-04-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080262036-A1 Phenyl-[1,2,4]-oxadiazol-5-one Derivatives, Pharmaceutical Compositions and Therapeutic Use Thereof GPR119, CPT1A, PC PPARA 87/4885PPARD 63/4885MDM2 3058/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.