SCHEMBL3783508

SCHEMBL3783508

c1cc2c(cc1N=C1NCCN1)CCC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.44
ADRA2B P18089 2/20 0.44
ADRA2C P18825 2/20 0.44
PNMT P11086 1/20 0.36
ALDH1A1 P00352 3/20 0.35
GRIN2D O15399 1/20 0.34
GRIN3B O60391 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2A Q12879 1/20 0.34
GRIN2B Q13224 1/20 0.34
GRIN2C Q14957 1/20 0.34
GRIN3A Q8TCU5 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA14 Q9ULX7 1/20 0.34
HPGD P15428 2/20 0.33
HSD17B10 Q99714 2/20 0.33
TSHR P16473 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3780069 0.96 ADRA2A (0.49) ADRA2AADRA2BADRA2CPNMTALDH1A1
SCHEMBL11184139 0.91 ADRA2A (0.47) ADRA2AADRA2BADRA2CPNMTALDH1A1
SCHEMBL16691804 0.75 ALDH1A1 (0.38) ALDH1A1HPGDHSD17B10GAA
SCHEMBL13063374 0.74 ADRA2A (0.52) ADRA2AADRA2BADRA2CALDH1A1GRIN2D
SCHEMBL22682041 0.70 ADRA2A (0.57) ADRA2AADRA2BADRA2CALDH1A1GRIN2D
SCHEMBL14404571 0.70 ADRA2A (0.52) ADRA2AADRA2BADRA2CPNMTALDH1A1
SCHEMBL9421173 0.69 PTGS1 (0.37) ALDH1A1CA1CA2HPGDHSD17B10
SCHEMBL12860178 0.67 ADRA2A (0.38) ADRA2AADRA2BADRA2CHPGDGAA
SCHEMBL3782607 0.66 HPGD (0.42) ALDH1A1HPGDHSD17B10GAARAB9A
SCHEMBL11215407 0.66 MAPT (0.44) ALDH1A1CA12CA2GAARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100331384-A1 GUANIDINE BASED COMPOUNDS UNIVERSIDAD DEL PAIS VASCO/EUSKAL HERRIKO UNIBERTSITATEA (ES) 2010-12-30 US disclosed
WO-2009080818-A2 GUANIDINE BASED COMPOUNDS THE PROVOST, FELLOWS AND SCHOLARS OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH NEAR DUBLIN (IE) 2009-07-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100331384-A1 GUANIDINE BASED COMPOUNDS ADRB2, ADRA2A, ADRA2C ADRA2A 2/4885ADRA2B 6/4885ADRA2C 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.