SCHEMBL3790649

SCHEMBL3790649

O=C(O)N1CCC(C(=O)O)(c2ccc(F)cc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.51
TET3 O43151 4/20 0.51
FBXL19 Q6PCT2 4/20 0.51
CXXC5 Q7LFL8 4/20 0.51
KDM2B Q8NHM5 4/20 0.51
CXXC4 Q9H2H0 4/20 0.51
KDM2A Q9Y2K7 4/20 0.51
TET1 Q8NFU7 3/20 0.51
HSD11B1 P28845 3/20 0.50
MLYCD O95822 1/20 0.48
APP P05067 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
OPRM1 P35372 1/20 0.46
AKR1C1 Q04828 1/20 0.44
S1PR2 O95136 2/20 0.43
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5171006 0.87 HSD11B1 (0.48) KMT2ATET3FBXL19CXXC5KDM2B
SCHEMBL23779147 0.84 KMT2A (0.69) KMT2ATET3FBXL19CXXC5KDM2B
SCHEMBL301150 0.84 APP (0.61) KMT2AHSD11B1MLYCDAPPCYP3A4
SCHEMBL3931269 0.83 KMT2A (0.71) KMT2ATET3FBXL19CXXC5KDM2B
SCHEMBL31292357 0.83 OPRM1 (0.63) KMT2ATET3FBXL19CXXC5KDM2B
SCHEMBL378380 0.82 SLC6A7 (0.54) KMT2ATET3FBXL19CXXC5KDM2B
Hydrochloric Acid SCHEMBL2772455 0.82 OPRM1 (0.66) KMT2ATET3FBXL19CXXC5KDM2B
SCHEMBL4728073 0.81 HSD11B1 (0.44) HSD11B1APPCYP3A4CYP2C9CYP2C19
SCHEMBL4725181 0.81 OPRM1 (0.55) CYP3A4OPRM1S1PR2
SCHEMBL378652 0.81 AKR1C3 (0.59) KMT2ATET3FBXL19CXXC5KDM2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010106081-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-23 WO disclosed