SCHEMBL4728073

SCHEMBL4728073

O=C(O)N1CCC(F)(c2ccc(F)cc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 8/20 0.44
CCR1 P32246 1/20 0.40
GRM5 P41594 1/20 0.40
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
CYP2C19 P33261 2/20 0.39
APP P05067 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
OPRM1 P35372 2/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
OPRL1 P41146 1/20 0.38
S1PR2 O95136 2/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12469550 0.86 HSD11B1 (0.46) HSD11B1GRM5OPRM1
SCHEMBL18711298 0.85 RORC (0.44) HSD11B1CYP2C19HTT
SCHEMBL4725181 0.83 OPRM1 (0.55) CCR1DRD2DRD4DRD3CYP3A4
SCHEMBL3790649 0.81 KMT2A (0.51) HSD11B1CYP2C19APPCYP3A4CYP2C9
SCHEMBL5807539 0.81 FASN (0.47)
SCHEMBL18701924 0.81 DRD2 (0.41) HSD11B1DRD2DRD4DRD3CYP2C19
Hydrochloric Acid SCHEMBL3428799 0.80 OPRM1 (0.52) CCR1DRD2DRD4DRD3CYP3A4
Hydrochloric Acid SCHEMBL3428801 0.80 OPRM1 (0.52) CCR1DRD2DRD4DRD3CYP3A4
SCHEMBL2425390 0.79 HSD11B1 (0.49) HSD11B1DRD2DRD4DRD3OPRM1
SCHEMBL1581427 0.79 OPRM1 (0.51) CCR1DRD2DRD4DRD3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008012623-A1 BENZIMIDAZOLYL COMPOUNDS AS POTENTIATORS OF MGLUR2 SUBTYPE OF GLUTAMATE RECEPTOR PFIZER PRODUCTS INC. (US) 2008-01-31 WO disclosed