SCHEMBL3795197

SCHEMBL3795197

N#Cc1cccc(-c2ccc(-c3[nH]c(-c4c(F)cccc4Cl)nc3Br)cn2)c1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGES O14684 12/20 0.47
GABRG2 P18507 2/20 0.38
GABRB3 P28472 2/20 0.38
GABRA5 P31644 2/20 0.38
GABRA3 P34903 2/20 0.38
KDM1A O60341 1/20 0.38
MAPK14 Q16539 1/20 0.38
JAK2 O60674 1/20 0.38
TYK2 P29597 1/20 0.38
HDAC2 Q92769 1/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2D6 P10635 1/20 0.37
IDO1 P14902 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3793065 0.91 PTGES (0.47) PTGESMAPK14JAK2TYK2CYP2C9
SCHEMBL13075515 0.87 PTGES (0.64) PTGESGABRG2GABRB3GABRA5GABRA3
SCHEMBL3790737 0.84 PTGES (0.49) PTGESKDM1AMAPK14CYP2C9
SCHEMBL3798464 0.81 PTGES (0.50) PTGESMAPK14CYP2C9CYP2D6
SCHEMBL3799359 0.80 PTGES (0.44) PTGESKDM1AMAPK14CYP2C9
SCHEMBL3805843 0.80 PTGES (0.46) PTGESMAPK14JAK2CYP2C9CYP2D6
SCHEMBL3799807 0.78 PTGES (0.43) PTGESMAPK14JAK2CYP2C9
SCHEMBL13075554 0.78 PTGES (0.64) PTGESMAPK14JAK2
SCHEMBL3796330 0.77 PTGES (0.41) PTGESMAPK14JAK2CYP2C9CYP2D6
SCHEMBL3795498 0.77 PTGES (0.45) PTGESMAPK14JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO claimed
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed