SCHEMBL3799359

SCHEMBL3799359

Fc1cccc(Cl)c1-c1nc(Br)c(-c2ccc(-c3ccc4sccc4c3)nc2)[nH]1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGES O14684 15/20 0.44
KDM1A O60341 1/20 0.39
ORAI1 Q96D31 2/20 0.37
CYP2C9 P11712 1/20 0.35
MAPK14 Q16539 1/20 0.35
PIK3CD O00329 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13076241 0.87 PTGES (0.55) PTGESKDM1AORAI1MAPK14PIK3CD
SCHEMBL3790737 0.81 PTGES (0.49) PTGESKDM1ACYP2C9MAPK14
SCHEMBL3795197 0.80 PTGES (0.47) PTGESKDM1ACYP2C9MAPK14
SCHEMBL3805843 0.79 PTGES (0.46) PTGESCYP2C9MAPK14
SCHEMBL3793065 0.79 PTGES (0.47) PTGESCYP2C9MAPK14
SCHEMBL3798464 0.79 PTGES (0.50) PTGESCYP2C9MAPK14
SCHEMBL3799807 0.77 PTGES (0.43) PTGESCYP2C9MAPK14
SCHEMBL3796330 0.77 PTGES (0.41) PTGESCYP2C9MAPK14
SCHEMBL3795498 0.75 PTGES (0.45) PTGESMAPK14
SCHEMBL3793346 0.73 MAPK14 (0.38) PTGESCYP2C9MAPK14PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO claimed
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed