SCHEMBL3795447

SCHEMBL3795447

O=C(NCc1ncccc1-c1ccc(F)cc1)c1ccc2n[nH]c(=O)n2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.43
ABL1 P00519 3/20 0.43
BCR P11274 3/20 0.43
PDPK1 O15530 2/20 0.41
CNR2 P34972 1/20 0.39
CNR1 P21554 1/20 0.38
NAMPT P43490 2/20 0.38
SLC40A1 Q9NP59 2/20 0.37
ADORA2A P29274 2/20 0.37
ADORA1 P30542 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
LIPG Q9Y5X9 1/20 0.36
DRD2 P14416 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3785444 0.85 NAMPT (0.44) AKT1ABL1BCRPDPK1NAMPT
SCHEMBL13258013 0.80 DRD2 (0.38) AKT1CNR2NAMPTSLC40A1ADORA2A
SCHEMBL13257863 0.80 AKT1 (0.37) AKT1CNR2NAMPTADORA2AADORA1
SCHEMBL13258147 0.78 LMNA (0.41) AKT1CNR1NAMPTMEN1KMT2A
SCHEMBL13075758 0.70 MAPT (0.45) CNR2CNR1KMT2A
SCHEMBL3790038 0.69 EPHX2 (0.52) HDAC3HDAC1HDAC2HDAC6
SCHEMBL13076485 0.68 GRIN1 (0.50) CNR2
SCHEMBL3793750 0.67 ROCK2 (0.57) NAMPTKMT2AHDAC1
SCHEMBL1870660 0.67 KMT2A (0.52) MEN1KMT2AHDAC6
SCHEMBL3789293 0.67 NAMPT (0.42) NAMPTADORA2AADORA1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010096722-A1 3-OXO-2, 3-DIHYDRO- [1,2, 4] TRIAZOLO [4, 3-A]PYRIDINES AS SOLUBLE EPOXIDE HYDROLASE (SEH) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-08-26 WO disclosed
WO-2010096722-A1 3-OXO-2, 3-DIHYDRO- [1,2, 4] TRIAZOLO [4, 3-A]PYRIDINES AS SOLUBLE EPOXIDE HYDROLASE (SEH) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-08-26 WO disclosed