SCHEMBL13258013

SCHEMBL13258013

O=C(NCc1ncccc1-c1ccc(F)cc1)c1ccc2nn(CCO)c(=O)n2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.38
AKT1 P31749 1/20 0.38
SLC40A1 Q9NP59 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
NAMPT P43490 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
ADORA2A P29274 5/20 0.36
CNR2 P34972 1/20 0.35
ADORA1 P30542 3/20 0.35
TP53 P04637 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
ADORA2B P29275 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13257863 0.90 AKT1 (0.37) DRD2AKT1MEN1KMT2ANAMPT
SCHEMBL13258147 0.88 LMNA (0.41) DRD2AKT1MEN1KMT2ANAMPT
SCHEMBL3789293 0.86 NAMPT (0.42) MEN1KMT2ANAMPTSMN1; SMN2ADORA2A
SCHEMBL3795447 0.80 AKT1 (0.43) DRD2AKT1SLC40A1MEN1KMT2A
SCHEMBL3789575 0.77 ALDH1A1 (0.40) MEN1KMT2ANAMPT
SCHEMBL3794645 0.76 NAMPT (0.42) MEN1KMT2ANAMPTSMN1; SMN2HDAC1
SCHEMBL3797563 0.74 NAMPT (0.43) MEN1KMT2ANAMPTSMN1; SMN2DGAT2
SCHEMBL3786760 0.72 EPHX2 (0.48) HDAC3HDAC1HDAC2HDAC6
SCHEMBL3789642 0.69 AKR1B1 (0.39)
SCHEMBL1870660 0.67 KMT2A (0.52) MEN1KMT2ATP53RXFP1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010096722-A1 3-OXO-2, 3-DIHYDRO- [1,2, 4] TRIAZOLO [4, 3-A]PYRIDINES AS SOLUBLE EPOXIDE HYDROLASE (SEH) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-08-26 WO disclosed