SCHEMBL3799989

SCHEMBL3799989

Fc1ccc(C2(c3nc(-c4ccc(-c5cnc(-c6c(F)cccc6Cl)[nH]5)cn4)no3)CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGES O14684 6/20 0.44
JAK2 O60674 1/20 0.36
HPGDS O60760 6/20 0.36
HSD11B1 P28845 1/20 0.34
NPC1 O15118 1/20 0.33
CASP3 P42574 1/20 0.33
RAB9A P51151 1/20 0.33
SENP8 Q96LD8 1/20 0.33
SENP7 Q9BQF6 1/20 0.33
SENP6 Q9GZR1 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
NPY5R Q15761 1/20 0.32
CHRNB2 P17787 2/20 0.31
CHRNA4 P43681 2/20 0.31
ADORA3 P0DMS8 1/20 0.31
REN P00797 1/20 0.31
CYP3A4 P08684 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13076381 0.87 HSD11B1 (0.34) PTGESJAK2HSD11B1NPC1CASP3
SCHEMBL3790517 0.80 PTGES (0.54) PTGESJAK2HPGDSNPC1CASP3
SCHEMBL3796009 0.80 PTGES (0.44) PTGESJAK2HPGDSNPC1RAB9A
SCHEMBL3803620 0.79 PTGES (0.43) PTGESJAK2HPGDSNPC1RAB9A
SCHEMBL3802070 0.79 PTGES (0.49) PTGESJAK2HPGDSNPC1CASP3
SCHEMBL3797930 0.78 PTGES (0.46) PTGESJAK2HPGDSHSD11B1NPC1
SCHEMBL3795318 0.78 PTGES (0.45) PTGESJAK2HPGDSNPC1CASP3
SCHEMBL3797347 0.77 PTGES (0.50) PTGESJAK2HPGDSNPC1RAB9A
SCHEMBL3794424 0.77 PTGES (0.47) PTGESJAK2HPGDSNPC1CASP3
SCHEMBL3793690 0.77 PTGES (0.46) PTGESJAK2HPGDSNPC1CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO claimed
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed