SCHEMBL3797019

SCHEMBL3797019

Fc1cccc(Cl)c1-c1ncc(C#Cc2cccc(C(F)(F)F)c2)[nH]1

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGES O14684 17/20 0.53
GRM5 P41594 1/20 0.41
PTGS1 P23219 1/20 0.40
SCN2A Q99250 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13075524 0.79 PTGES (0.57) PTGESGRM5PTGS1
SCHEMBL3794537 0.77 PTGES (0.54) PTGESGRM5PTGS1
SCHEMBL3798131 0.73 PTGES (0.43) PTGES
SCHEMBL3795873 0.73 PTGES (0.49) PTGES
SCHEMBL12478777 0.70 PTGES (0.77) PTGESPTGS1
SCHEMBL2361302 0.70 PTGES (0.58) PTGES
SCHEMBL30873473 0.68 GRM5 (0.58) PTGESGRM5
SCHEMBL3800830 0.67 PTGES (0.54) PTGESPTGS1SCN2A
SCHEMBL3799817 0.66 PDE4A (0.39) PTGES
SCHEMBL1476835 0.65 CHRNB2 (0.51) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO claimed