SCHEMBL3798547

SCHEMBL3798547

COC(=O)c1ccc2cc(-c3c[nH]c(-c4c(F)cccc4Cl)n3)oc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 4/20 0.39
MAPK14 Q16539 2/20 0.38
RHEB Q15382 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
PSMB8 P28062 1/20 0.36
APP P05067 1/20 0.35
HPGD P15428 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TP53 P04637 2/20 0.35
MAPT P10636 2/20 0.35
CREBBP Q92793 1/20 0.34
PIM1 P11309 1/20 0.34
CSNK2A2 P19784 1/20 0.34
CSNK2B P67870 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3790901 0.93 PTGES (0.39) PTGESMAPK14RHEBNPC1RAB9A
SCHEMBL3797090 0.88 RHEB (0.41) PTGESMAPK14RHEBNPC1RAB9A
SCHEMBL4784907 0.81 RHEB (0.46) PTGESMAPK14RHEBNPC1RAB9A
SCHEMBL3792228 0.81 PTGES (0.39) PTGESAPPTP53MAPTPIM1
SCHEMBL3800146 0.74 PIM1 (0.49) PTGESNPC1RAB9APIM1CSNK2A2
SCHEMBL3795502 0.73 PTGES (0.43) PTGESPIM1CSNK2A2CSNK2BPIM3
SCHEMBL3796734 0.73 PTGES (0.43) PTGESPIM1CSNK2A2CSNK2BPIM3
SCHEMBL3802320 0.72 PTGES (0.40) PTGESPIM1CSNK2A2CSNK2BPIM3
SCHEMBL3791130 0.71 PTGES (0.42) PTGESPIM1CSNK2A2CSNK2BPIM3
SCHEMBL2362023 0.71 RHEB (0.57) PTGESMAPK14RHEBNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO claimed
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed