SCHEMBL3801397

SCHEMBL3801397

COc1ccc(CC(C)(C)C(=O)O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.53
PPARA Q07869 2/20 0.50
HTT P42858 1/20 0.49
MMP1 P03956 2/20 0.48
MMP13 P45452 2/20 0.48
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
POLB P06746 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CTBP2 P56545 1/20 0.47
F2RL1 P55085 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CYP4F2 P78329 1/20 0.46
CYP4A11 Q02928 1/20 0.46
PPARG P37231 1/20 0.46
MMP9 P14780 1/20 0.46
LTA4H P09960 1/20 0.46
FFAR1 O14842 1/20 0.45
MEN1 O00255 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4413232 0.98 LDHA (0.51) LDHAPPARAHTTMMP1MMP13
SCHEMBL28246723 0.98 LDHA (0.51) LDHAPPARAHTTMMP1MMP13
SCHEMBL20269317 0.85 SMN1; SMN2 (0.49) LDHAHTTMMP1MMP13NPC1
SCHEMBL28136422 0.85 LDHA (0.53) LDHAPPARAHTTMMP1MMP13
SCHEMBL7676911 0.84 LDHA (0.51) LDHAPPARAHTTMMP1MMP13
SCHEMBL13903099 0.84 PTPRB (0.54) LDHAHTTMMP1MMP13NPC1
SCHEMBL3739737 0.84 LDHA (0.51) LDHAPPARAHTTMMP1MMP13
SCHEMBL5208103 0.83 LDHA (0.55) LDHAHTTNPC1RAB9APOLB
SCHEMBL1424653 0.82 BLM (0.67) LDHAPPARAHTTMMP1MMP13
SCHEMBL2033365 0.82 BLM (0.67) LDHAPPARAHTTMMP1MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230046065-A1 MERGING C(sp3)-H ACTIVATION WITH DNA-ENCODING THE SCRIPPS RESEARCH INSTITUTE 2023-02-16 US disclosed
CN-108586500-A Zinc co-ordination complex and the method for preparing organic zinc reagent 慕尼黑路德维希马克西米利安斯大学 2018-09-28 CN disclosed
CN-103429598-B Organozinc complexes and methods of making and using the same 慕尼黑路德维希马克西米利安斯大学 2018-03-30 CN disclosed
EP-2065360-B1 Use of 3-methylbenzyl isobutyrate as a fragrance compound SYMRISE AG (DE) 2013-06-19 EP disclosed
US-7902394-B2 Calcilytic compounds GLAXOSMITHKLINE LLC (US) 2011-03-08 US disclosed
US-20100029782-A1 Calcilytic Compounds SMITHKLINE BEECHAM CORPORATION (US) 2010-02-04 US disclosed
EP-2120898-A1 CALCILYTIC COMPOUNDS SmithKline Beecham Corporation (US) 2009-11-25 EP disclosed
EP-2065360-A2 3-methylbenzyl isobutyrate Symrise GmbH & Co. KG (DE) 2009-06-03 EP disclosed
EP-1747186-B1 Fragrant composition comprising 3-methylbenzyl-isobutyrat SYMRISE GMBH & CO KG (DE) 2009-03-11 EP disclosed
WO-2008077009-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-06-26 WO disclosed
CN-1221401-A Calcilytic compounds NPS PHARMA INC (US) 1999-06-30 CN disclosed
EP-0901459-A1 CALCILYTIC COMPOUNDS NPS PHARMACEUTICALS, INC. (US) 1999-03-17 EP disclosed
WO-1997037967-A1 CALCILYTIC COMPOUNDS NPS PHARMACEUTICALS, INC. (US) 1997-10-16 WO disclosed
EP-0421759-B1 Method for producing 1-indanone derivatives HOECHST CELANESE CORP (US) 1995-06-07 EP disclosed
US-5179229-A Preparation of 2,2-diorgano-3-arylpropionic acids and esters thereof HOECHST CELANESE CORPORATION (US) 1993-01-12 US disclosed
US-5012007-A Method for producing 1-indanone derivatives HOECHST CELANESE CORPORATION, A CORP. OF DE 1991-04-30 US disclosed
EP-0421759-A2 Method for producing 1-indanone derivatives HOECHST CELANESE CORPORATION (US) 1991-04-10 EP disclosed
US-4898608-A Pyridylthio-acylanilide herbicides BAYER AKTIENGESELLSCHAFT (DE) 1990-02-06 US disclosed
US-4797146-A INSECTICIDES, FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 1989-01-10 US disclosed
US-4627871-A Herbicidal 2-[4-substituted carboxyamino-phenoxy (or phenyl mercapto)]-substituted pyrimidines BAYER AKTIENGESELLSCHAFT (DE) 1986-12-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100029782-A1 Calcilytic Compounds CALCR, CALCA, CALCB LDHA 3727/4885PPARA 3735/4885HTT 4483/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.