SCHEMBL3816899

SCHEMBL3816899

NNC1CCN(CC2c3ccccc3-c3ccccc32)CC1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.42
ACHE P22303 4/20 0.37
CCR1 P32246 3/20 0.36
BCHE P06276 3/20 0.36
BACE1 P56817 2/20 0.36
HTR2C P28335 2/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
UBE2M P61081 1/20 0.34
DCUN1D1 Q96GG9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21995339 0.79 ACHE (0.52) HTR2AACHESIGMAR1
SCHEMBL28397007 0.78 HTR2A (0.47) HTR2A
SCHEMBL29575598 0.76 METAP1 (0.49) HTR2A
SCHEMBL1119003 0.76 METAP1 (0.49) HTR2A
SCHEMBL1128712 0.74 KMT2A (0.48)
SCHEMBL295894 0.73 L3MBTL1 (0.49) HTR2AHTR2CCA1CA2SIGMAR1
SCHEMBL15688648 0.73 SIGMAR1 (0.46) HTR2AHTR2CSIGMAR1
SCHEMBL875259 0.73 HTR2C (0.44) HTR2AHTR2C
SCHEMBL117304 0.70 ACHE (0.68) HTR2AACHEBCHEBACE1HTR2C
SCHEMBL19183445 0.70 HTR2A (0.43) HTR2ACA1CA2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765805-A4 CGRP RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2009-08-26 EP disclosed
EP-1765805-A2 CGRP RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2007-03-28 EP disclosed
WO-2005072308-A2 CGRP RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2005-08-11 WO disclosed