SCHEMBL3824652

SCHEMBL3824652

COc1cccc(-c2nc(C)oc2C(N)=O)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.55
RIPK2 O43353 1/20 0.48
PARP1 P09874 2/20 0.47
SLC9A1 P19634 1/20 0.46
RXRA P19793 1/20 0.45
RXRB P28702 1/20 0.45
PIN1 Q13526 1/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.44
KDM4E B2RXH2 4/20 0.44
HSD17B10 Q99714 2/20 0.44
LMNA P02545 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MAPT P10636 1/20 0.44
ADORA3 P0DMS8 2/20 0.43
ADORA2B P29275 2/20 0.43
ADORA1 P30542 2/20 0.43
ADORA2A P29274 2/20 0.43
PLG P00747 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3822883 0.83 RIPK2 (0.46) RIPK2PARP1SLC9A1RXRARXRB
SCHEMBL3826031 0.81 SLC9A1 (0.44) PARP1SLC9A1ALDH1A1KDM4EADORA1
SCHEMBL5008392 0.80 KDM4E (0.58) IKBKBALDH1A1KDM4EHSD17B10LMNA
SCHEMBL3822654 0.77 KDM4E (0.55) IKBKBRXRARXRBALDH1A1KDM4E
SCHEMBL3824657 0.76 DPP4 (0.51) IKBKBALDH1A1HPGDKDM4EHSD17B10
Hydrochloric Acid SCHEMBL3825192 0.75 DPP4 (0.50) IKBKBALDH1A1HPGDKDM4EHSD17B10
SCHEMBL3823644 0.74 IKBKB (0.49) IKBKBPARP1RXRARXRBALDH1A1
SCHEMBL1167406 0.72 PIN1 (0.57) IKBKBRXRARXRBPIN1ALDH1A1
SCHEMBL13312255 0.72 SMN1; SMN2 (0.47) IKBKBRXRARXRBALDH1A1HPGD
SCHEMBL3826511 0.72 IKBKB (0.47) IKBKBALDH1A1KDM4EHSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2096111-A1 PYRAZOLES AND USE THEREOF AS DRUGS Japan Tobacco Inc. (JP) 2009-09-02 EP claimed
US-20090036450-A1 PYRAZOLE COMPOUNDS AND USE THEREOF JAPAN TOBACCO, INC. (JP) 2009-02-05 US claimed
US-20090036450-A1 PYRAZOLE COMPOUNDS AND USE THEREOF JAPAN TOBACCO, INC. (JP) 2009-02-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090036450-A1 PYRAZOLE COMPOUNDS AND USE THEREOF PYGL, GYS2, G6PC1 IKBKB 1573/4885RIPK2 2526/4885PARP1 2289/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.