SCHEMBL3825935

SCHEMBL3825935

NC(=O)c1nnc(-c2cccc(Cl)c2)[nH]1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.54
PIN1 Q13526 1/20 0.48
HRH1 P35367 1/20 0.48
NUDT1 P36639 1/20 0.46
SLC9A1 P19634 1/20 0.45
IKBKB O14920 3/20 0.45
IDO1 P14902 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
CHUK O15111 1/20 0.43
GAA P10253 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MPI P34949 1/20 0.42
GFER P55789 1/20 0.42
JAK2 O60674 1/20 0.42
TYMP P19971 1/20 0.41
MGAM O43451 1/20 0.40
SI P14410 1/20 0.40
MGAM2 Q2M2H8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4013450 0.80 NPC1 (0.49) PARP1PIN1NPC1RAB9A
SCHEMBL3825940 0.74 HRH1 (0.56) PARP1PIN1HRH1IDO1NPC1
SCHEMBL11486446 0.74 PIN1 (0.59) PARP1PIN1HRH1NUDT1SLC9A1
SCHEMBL12128300 0.72 PIN1 (0.48) PARP1PIN1HRH1IDO1GAA
SCHEMBL31429182 0.72 HRH1 (0.50) PARP1PIN1HRH1IDO1NPC1
SCHEMBL416660 0.72 GAA (0.53) PIN1HRH1IDO1GAAKDM4E
SCHEMBL15330500 0.72 HRH1 (0.47) PARP1PIN1HRH1IDO1NPC1
SCHEMBL3726438 0.71 PARP1 (0.50) PARP1PIN1NUDT1IKBKBNPC1
SCHEMBL12128291 0.71 PIN1 (0.47) PARP1PIN1HRH1SLC9A1IDO1
SCHEMBL29412056 0.71 PARP1 (1.00) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2096111-A1 PYRAZOLES AND USE THEREOF AS DRUGS Japan Tobacco Inc. (JP) 2009-09-02 EP disclosed
US-20090036450-A1 PYRAZOLE COMPOUNDS AND USE THEREOF JAPAN TOBACCO, INC. (JP) 2009-02-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090036450-A1 PYRAZOLE COMPOUNDS AND USE THEREOF PYGL, GYS2, G6PC1 PARP1 2289/4885PIN1 1595/4885HRH1 4618/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.