SCHEMBL3826441

SCHEMBL3826441

O=C(c1ccc(Cl)cc1)N(Cc1ccc(NC2CC2)nc1)c1ccc(F)cc1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.49
BCL2A1 Q16548 1/20 0.45
KCNQ3 O43525 1/20 0.43
KCNQ2 O43526 1/20 0.43
VNN1 O95497 1/20 0.43
PRKAA2 P54646 1/20 0.43
HCAR3 P49019 3/20 0.43
PDK1 Q15118 4/20 0.42
PDK2 Q15119 2/20 0.39
PDK4 Q16654 2/20 0.39
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
PDK3 Q15120 1/20 0.39
KCNH2 Q12809 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3828503 0.87 IKBKB (0.45) MAPK14BCL2A1VNN1PDK1
SCHEMBL3823686 0.86 BCL2A1 (0.47) MAPK14BCL2A1VNN1HCAR3PDK1
SCHEMBL3829758 0.84 BCL2A1 (0.45) MAPK14BCL2A1VNN1PDK1PDK2
SCHEMBL3822748 0.82 BCL2A1 (0.52) MAPK14BCL2A1KCNQ3KCNQ2VNN1
SCHEMBL4735448 0.81 MAPK14 (0.55) MAPK14HCAR3PDK1
SCHEMBL3058152 0.80 CYP11B1 (0.43) MAPK14KCNQ3KCNQ2VNN1PRKAA2
SCHEMBL3828507 0.80 PDK1 (0.45) MAPK14BCL2A1VNN1PDK1PDK2
SCHEMBL3830084 0.79 PDK1 (0.49) MAPK14BCL2A1VNN1PDK1PDK2
SCHEMBL3824490 0.79 MCHR1 (0.47) PRKAA2KCNH2
SCHEMBL4737583 0.79 GAA (0.46) MAPK14PDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2097379-A1 CARBOXAMIDE DERIVATIVES AS ION CHANNEL MODULATORS Wyeth a Corporation of the State of Delaware (US) 2009-09-09 EP claimed
WO-2008073936-A1 CARBOXAMIDE DERIVATIVES AS ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed