SCHEMBL3828503

SCHEMBL3828503

O=C(c1ccc(Cl)cc1)N(Cc1ccc(NCC2CC2)nc1)c1ccc(F)cc1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 4/20 0.45
CRHR1 P34998 4/20 0.44
BCL2A1 Q16548 1/20 0.43
VNN1 O95497 1/20 0.41
PDK1 Q15118 1/20 0.40
MAPK14 Q16539 4/20 0.40
GABRA5 P31644 1/20 0.39
ACHE P22303 1/20 0.38
CCNK O75909 1/20 0.38
CDK9 P50750 1/20 0.38
S1PR1 P21453 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3826441 0.87 MAPK14 (0.49) BCL2A1VNN1PDK1MAPK14
SCHEMBL3829758 0.85 BCL2A1 (0.45) BCL2A1VNN1PDK1MAPK14
SCHEMBL3823686 0.84 BCL2A1 (0.47) BCL2A1VNN1PDK1MAPK14
SCHEMBL3058766 0.81 CRHR1 (0.45) IKBKBCRHR1VNN1GABRA5ACHE
SCHEMBL3822748 0.80 BCL2A1 (0.52) BCL2A1VNN1PDK1MAPK14
SCHEMBL3828507 0.78 PDK1 (0.45) BCL2A1VNN1PDK1MAPK14
SCHEMBL3830084 0.77 PDK1 (0.49) BCL2A1VNN1PDK1MAPK14
SCHEMBL3829755 0.76 PDK1 (0.48) BCL2A1VNN1PDK1MAPK14
SCHEMBL3831162 0.75 RAB9A (0.53) BCL2A1PDK1MAPK14
SCHEMBL3821700 0.75 CNR2 (0.49) BCL2A1VNN1PDK1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2097379-A1 CARBOXAMIDE DERIVATIVES AS ION CHANNEL MODULATORS Wyeth a Corporation of the State of Delaware (US) 2009-09-09 EP claimed
WO-2008073936-A1 CARBOXAMIDE DERIVATIVES AS ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed