SCHEMBL383152

SCHEMBL383152

COc1ccccc1[C](c1ccccc1OC)c1cccc2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.51
ALDH1A1 P00352 2/20 0.51
HTT P42858 1/20 0.51
MAPT P10636 2/20 0.48
ESR1 P03372 1/20 0.46
ESR2 Q92731 1/20 0.46
KMT2A Q03164 3/20 0.46
GAA P10253 1/20 0.46
CACNA1B Q00975 1/20 0.46
APBA1 Q02410 1/20 0.46
AKR1C2 P52895 1/20 0.46
NR4A1 P22736 1/20 0.46
NR4A2 P43354 1/20 0.46
NR4A3 Q92570 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
MEN1 O00255 2/20 0.45
PLK1 P53350 1/20 0.44
CNR2 P34972 2/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL157181 0.84 CA1 (0.60) HTTKMT2AGAAMEN1RAB9A
SCHEMBL9856908 0.82 CDC25B (0.59) POLBALDH1A1HTTESR1ESR2
SCHEMBL2494543 0.82 NR4A1 (0.62) POLBALDH1A1MAPTKMT2AGAA
SCHEMBL151449 0.78 MAPT (0.61) ALDH1A1MAPTKMT2AGAAL3MBTL1
SCHEMBL29367279 0.78 MAPT (0.61) ALDH1A1MAPTKMT2AGAAL3MBTL1
SCHEMBL30373629 0.78 MAPT (0.61) ALDH1A1MAPTKMT2AGAAL3MBTL1
SCHEMBL3854662 0.77 KMT2A (0.53) POLBALDH1A1HTTMAPTKMT2A
SCHEMBL3862642 0.77 KMT2A (0.53) POLBALDH1A1HTTMAPTKMT2A
SCHEMBL31321659 0.76 KMT2A (0.69) POLBALDH1A1HTTMAPTESR1
1,2-Dimethoxybenzene SCHEMBL20581614 0.76 CA12 (0.62) ALDH1A1HTTMAPTKMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 191 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140142253-A1 Dithiolane Based Thiol Modifier For Labeling and Stronger Immobilization of Bio-Molecules On Solid Surfaces CHEMGENES CORPORATION (US) 2014-05-22 US claimed
US-8541569-B2 Phosphoramidites for synthetic RNA in the reverse direction, efficient RNA synthesis and convenient introduction of 3'-end ligands, chromophores and modifications of synthetic RNA CHEMGENES CORPORATION (US) 2013-09-24 US claimed
WO-2013126034-A1 SYNTHESIS OF HIGH PURITY DMT-C3-DISULFIDE PHOSPHORAMIDITE CHEMGENES CORPORATION (US) 2013-08-29 WO claimed
EP-2560982-A2 PHOSPHORAMIDITES FOR SYNTHETIC RNA IN THE REVERSE DIRECTION Chemgenes Corporation (US) 2013-02-27 EP claimed
WO-2011103468-A2 PHOSPHORAMIDITES FOR SYNTHETIC RNA IN THE REVERSE DIRECTION CHEMGENES CORPORATION (US) 2011-08-25 WO claimed
US-20110137010-A1 PHOSPHORAMIDITES FOR SYNTHETIC RNA IN THE REVERSE DIRECTION, EFFICIENT RNA SYNTHESIS AND CONVENIENT INTRODUCTION OF 3'-END LIGANDS, CHROMOPHORES AND MODIFICATIONS OF SYNTHETIC RNA CHEMGENES CORPORATION (US) 2011-06-09 US claimed
EP-2121719-A2 2-5A DERIVATIVES AND THEIR USE AS ANTI-CANCER, ANTI-VIRAL AND ANTI-PARASITIC AGENTS Alios Biopharma, Inc. (US) 2009-11-25 EP claimed
WO-2009086192-A1 BIODEGRADABLE PHOSPHATE PROTECTED NUCLEOTIDE DERIVATIVES AND THEIR USE AS CANCER, ANTI VIRAL AND ANTI PARASITIC AGENTS ALIOS BIOPHARMA, INC. (US) 2009-07-09 WO claimed
WO-2009086201-A1 2-5A ANALOGS AND THEIR USE AS ANTI-CANCER, ANTI-VIRAL AND ANTI- PARAS ITI C AGENTS ALIOS BIOPHARMA, INC. (US) 2009-07-09 WO claimed
WO-2008095040-A2 2-5A DERIVATIVES AND THEIR USE AS ANTI-CANCER, ANTI-VIRAL AND ANTI-PARASITIC AGENTS ALIOS BIOPHARMA, INC. (US) 2008-08-07 WO claimed
US-6239220-B1 Recovery of triarylmethyl halide protecting groups cleaved during oligonucleotide synthesis ISIS PHARMACEUTICALS, INC. 2001-05-29 US claimed
US-6124484-A Recovery of triarylmethyl halide protecting groups cleaved during oligonucleotide synthesis ISIS PHARMACEUTICALS, INC. (US) 2000-09-26 US claimed
WO-2000004062-A1 RECOVERY OF TRIARYLMETHYL HALIDE PROTECTING GROUPS CLEAVED DURING OLIGONUCLEOTIDE SYNTHESIS ISIS PHARMACEUTICALS, INC. (US) 2000-01-27 WO claimed
US-4668777-A POLYNUCLEOTIDE INTERMEDIATES UNIVERSITY PATENTS, INC. (US) 1987-05-26 US claimed
EP-0061746-B1 PHOSPHORAMIDITE COMPOUNDS AND THEIR USE IN PRODUCING OLIGONUCLEOTIDES UNIVERSITY PATENTS, INC. (US) 1985-03-20 EP claimed
CN-117379452-A Substituted nucleosides, nucleotides and analogues thereof 艾丽奥斯生物制药有限公司 2024-01-12 CN disclosed
EP-3160475-B1 SUBSTITUTED NUCLEOSIDES AND NUCLEOTIDES TO TREAT FILOVIRIDAE INFECTIONS JANSSEN PHARMACEUTICALS INC (US) 2024-01-03 EP disclosed
EP-0144386-A1 NOVEL PREPARATION OF NUCLEOSIDE PHOSPHORAMIDITE INTERMEDIATES. BECKMAN INSTRUMENTS INC (US) 1985-06-19 EP disclosed
WO-1984004749-A1 NOVEL PREPARATION OF NUCLEOSIDE PHOSPHORAMIDITE INTERMEDIATES BECKMAN INSTRUMENTS INC (US) 1984-12-06 WO disclosed
EP-0061746-A1 Phosphoramidite compounds and their use in producing oligonucleotides UNIVERSITY PATENTS, INC. (US) 1982-10-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140142253-A1 Dithiolane Based Thiol Modifier For Labeling and Stronger Immobilization of Bio-Molecules On Solid Surfaces PTMS, SPOUT1, SRMS POLB 83/4885ALDH1A1 1329/4885HTT 4109/4885
US-20110137010-A1 PHOSPHORAMIDITES FOR SYNTHETIC RNA IN THE REVERSE DIRECTION, EFFICIENT RNA SYNTHESIS AND CONVENIENT INTRODUCTION OF 3'-END LIGANDS, CHROMOPHORES AND MODIFICATIONS OF SYNTHETIC RNA NSUN3, RNGTT, NOP2 POLB 48/4885ALDH1A1 4050/4885HTT 2036/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.